Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50007699
TargetCoagulation factor X(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17277(CHEMBL55035 | 4-{[(1Z,3Z)-3-[(4-carbamimidoylpheny...)
Affinity DataKi:  0.660nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066616(2,7-di[1-[3-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  5.60nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066615(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  29nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17277(CHEMBL55035 | 4-{[(1Z,3Z)-3-[(4-carbamimidoylpheny...)
Affinity DataKi:  33nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066616(2,7-di[1-[3-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  44nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066615(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  130nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066613((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  140nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066613((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  200nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066615(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  200nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066614(2,7-di[1-[4-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  280nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066612(2,7-di[1-[3-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  410nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17277(CHEMBL55035 | 4-{[(1Z,3Z)-3-[(4-carbamimidoylpheny...)
Affinity DataKi:  530nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066613((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  1.00E+3nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066612(2,7-di[1-[3-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  1.40E+3nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066616(2,7-di[1-[3-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  1.40E+3nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066612(2,7-di[1-[3-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  2.10E+3nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066614(2,7-di[1-[4-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  6.20E+3nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066614(2,7-di[1-[4-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  1.70E+4nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed