Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 5179
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50021325(DIHYDROMORPHINE | CHEMBL1281 | 4-methyl-(1S,5R,13R...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50003571(17-methyl-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]...)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50003571(17-methyl-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]...)
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50021325(DIHYDROMORPHINE | CHEMBL1281 | 4-methyl-(1S,5R,13R...)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  1.16nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  1.29nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50016847(CHEMBL337041 | Cyprodime)
Affinity DataKi:  4.59nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50016847(CHEMBL337041 | Cyprodime)
Affinity DataKi:  7.23nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50018708(DSLET-OH | DSLET | CHEMBL124283 | Tyr-D-Ser-Gly-Ph...)
Affinity DataKi:  7.34nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50018708(DSLET-OH | DSLET | CHEMBL124283 | Tyr-D-Ser-Gly-Ph...)
Affinity DataKi:  8.71nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  10.8nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  25.7nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21130(U69,593 | N-methyl-N-(7-(1-pyrrolidinyl)-1-oxaspir...)
Affinity DataKi:  253nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50003571(17-methyl-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]...)
Affinity DataKi:  539nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21130(U69,593 | N-methyl-N-(7-(1-pyrrolidinyl)-1-oxaspir...)
Affinity DataKi:  591nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  707nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50003571(17-methyl-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]...)
Affinity DataKi:  779nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  1.01E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50041958(TIPP | CHEMBL108731 | 2-[1-{2-[2-amino-3-(4-hydrox...)
Affinity DataKi:  1.71E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50057010((S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  2.52E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50041958(TIPP | CHEMBL108731 | 2-[1-{2-[2-amino-3-(4-hydrox...)
Affinity DataKi:  9.15E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed