Compile Data Set for Download or QSAR
Report error Found 189 Enz. Inhib. hit(s) with all data for entry = 50003489
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471700(CHEMBL91022)
Affinity DataKi:  0.229nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50366618(SNAP-5089 | CHEMBL448620)
Affinity DataKi:  0.347nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471684(CHEMBL327931)
Affinity DataKi:  0.525nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50068828(2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataKi:  1nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50068828(2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataKi:  1nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471694(CHEMBL91550)
Affinity DataKi:  1.10nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471697(CHEMBL91415)
Affinity DataKi:  1.10nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471698(CHEMBL89685)
Affinity DataKi:  1.20nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471696(CHEMBL315914)
Affinity DataKi:  1.40nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471685(CHEMBL313160)
Affinity DataKi:  1.5nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471692(CHEMBL89243)
Affinity DataKi:  1.80nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471695(CHEMBL314960)
Affinity DataKi:  1.80nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471687(CHEMBL327712)
Affinity DataKi:  1.90nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471703(CHEMBL284103)
Affinity DataKi:  4.5nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  6.90nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471701(CHEMBL315538)
Affinity DataKi:  7.10nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471691(CHEMBL312871)
Affinity DataKi:  8.70nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471706(CHEMBL91956)
Affinity DataKi:  8.70nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471690(CHEMBL88388)
Affinity DataKi:  8.90nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471700(CHEMBL91022)
Affinity DataKi:  13nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471686(CHEMBL284470)
Affinity DataKi:  15nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471689(CHEMBL88628)
Affinity DataKi:  16nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471702(CHEMBL88448)
Affinity DataKi:  20nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50068828(2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataKi:  20.9nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  31nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471693(CHEMBL92322)
Affinity DataKi:  36nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471684(CHEMBL327931)
Affinity DataKi:  42nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471684(CHEMBL327931)
Affinity DataKi:  48nMAssay Description:Binding affinity assayed by displacement of [3H]rauwolscine from human alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471705(CHEMBL313953)
Affinity DataKi:  54nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471699(CHEMBL327775)
Affinity DataKi:  56nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471704(CHEMBL315392)
Affinity DataKi:  59nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471700(CHEMBL91022)
Affinity DataKi:  66nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471706(CHEMBL91956)
Affinity DataKi:  78nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471700(CHEMBL91022)
Affinity DataKi:  81nMAssay Description:Binding affinity assayed by displacement of [3H]rauwolscine from human alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471684(CHEMBL327931)
Affinity DataKi:  91nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471684(CHEMBL327931)
Affinity DataKi:  110nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471687(CHEMBL327712)
Affinity DataKi:  115nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471695(CHEMBL314960)
Affinity DataKi:  123nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471684(CHEMBL327931)
Affinity DataKi:  126nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471686(CHEMBL284470)
Affinity DataKi:  135nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471693(CHEMBL92322)
Affinity DataKi:  138nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50068828(2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataKi:  151nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50068828(2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataKi:  151nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471692(CHEMBL89243)
Affinity DataKi:  151nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471687(CHEMBL327712)
Affinity DataKi:  158nMAssay Description:Binding affinity assayed by displacement of [3H]rauwolscine from human alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471685(CHEMBL313160)
Affinity DataKi:  162nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50471705(CHEMBL313953)
Affinity DataKi:  162nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50068828(2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataKi:  165nMAssay Description:Binding affinity assayed by displacement of [3H]rauwolscine from human alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
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