Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 5153
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(NSC_5311134 | CAS_5311134 | GR 196429)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(NSC_5311134 | CAS_5311134 | GR 196429)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(NSC_5311134 | CAS_5311134 | GR 196429)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM82509(melatonin, 6-Hydroxy | Melatonin,6-Hydroxy)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(NSC_5311134 | CAS_5311134 | GR 196429)
Affinity DataKi:  0.610nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM82509(melatonin, 6-Hydroxy | Melatonin,6-Hydroxy)
Affinity DataKi:  1.69nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM82509(melatonin, 6-Hydroxy | Melatonin,6-Hydroxy)
Affinity DataKi:  2.23nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  2.69nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM82509(melatonin, 6-Hydroxy | Melatonin,6-Hydroxy)
Affinity DataKi:  10.2nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85065(CAS_117946-91-5 | NSC_122162 | Luzindole)
Affinity DataKi:  14.4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM82509(melatonin, 6-Hydroxy | Melatonin,6-Hydroxy)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29612(N-Acetyltryptamine,5-Hydroxy | CHEMBL33103 | Norme...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29612(N-Acetyltryptamine,5-Hydroxy | CHEMBL33103 | Norme...)
Affinity DataKi:  148nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85065(CAS_117946-91-5 | NSC_122162 | Luzindole)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85065(CAS_117946-91-5 | NSC_122162 | Luzindole)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1B(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29612(N-Acetyltryptamine,5-Hydroxy | CHEMBL33103 | Norme...)
Affinity DataKi:  302nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29612(N-Acetyltryptamine,5-Hydroxy | CHEMBL33103 | Norme...)
Affinity DataKi:  347nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29612(N-Acetyltryptamine,5-Hydroxy | CHEMBL33103 | Norme...)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85065(CAS_117946-91-5 | NSC_122162 | Luzindole)
Affinity DataKi:  676nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMelatonin receptor type 1A(Pig)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85065(CAS_117946-91-5 | NSC_122162 | Luzindole)
Affinity DataKi:  933nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed