Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50007533
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064365(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 0.400nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064373(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 0.600nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064359(1,18-Dihydroxy-12-[2-(4-hydroxy-3-methoxy-cyclohex...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064361(N-Cyclohexyl-2-{4-[2-(17-ethyl-1,14-dihydroxy-23,2...)
Affinity DataIC50: 2nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50068939(CHEMBL8597 | 17-Ethyl-1,14-dihydroxy-12-[2-(4-hydr...)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064375(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 2.40nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064355((E)-(1R,9S,12S,13R,14S,17R,21S,23S,25S,27R)-17-All...)
Affinity DataIC50: 2.5nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064374(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064351(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 3.20nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064350(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 3.30nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064353({4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-13,...)
Affinity DataIC50: 4nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064352(N-Benzyl-2-{4-[2-(17-ethyl-1,14-dihydroxy-23,25-di...)
Affinity DataIC50: 5.60nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064362({4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-13,...)
Affinity DataIC50: 9.40nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064363(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 13nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064376(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 16nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064367(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 19nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064357(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 46nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064358(N-Benzyl-2-{4-[2-(17-ethyl-1,14-dihydroxy-23,25-di...)
Affinity DataIC50: 48nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064369(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 50nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064360({4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-13,...)
Affinity DataIC50: 68nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064364(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 71nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064371(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 170nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064372(N-(4-Chloro-phenyl)-2-{4-[2-(17-ethyl-1,14-dihydro...)
Affinity DataIC50: 180nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064368(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 180nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064370(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 470nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064354(N-(3,4-Dichloro-phenyl)-2-{4-[2-(17-ethyl-1,14-dih...)
Affinity DataIC50: 500nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50064366(2-{4-[2-(17-Ethyl-1,14-dihydroxy-23,25-dimethoxy-1...)
Affinity DataIC50: 570nMAssay Description:Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails Article
PubMed