Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50036703
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062860(N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-y...)
Affinity DataIC50: 2.40nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062871(Pentanoic acid ({[3-(3-bromo-2-methyl-imidazo[1,2-...)
Affinity DataIC50: 7.80nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062878(N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-y...)
Affinity DataIC50: 8.90nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062864(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 9nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062863(CHEMBL154188 | 2-Acetylamino-N-[3-(3-bromo-2-methy...)
Affinity DataIC50: 16nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062863(CHEMBL154188 | 2-Acetylamino-N-[3-(3-bromo-2-methy...)
Affinity DataIC50: 16nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062865(N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-y...)
Affinity DataIC50: 19nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062898(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 26nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062905(3-Bromo-8-(2,6-dichloro-3-nitro-benzyloxy)-2-methy...)
Affinity DataIC50: 42nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062899(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 46nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062891(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 54nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062868(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 72nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062901(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 150nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062893(3-Chloro-8-(2,6-dichloro-benzyloxy)-2-methyl-imida...)
Affinity DataIC50: 200nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062884(3-Bromo-8-(2,6-dichloro-benzyloxy)-2-methyl-imidaz...)
Affinity DataIC50: 230nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062890(1-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 350nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062867(2-Amino-N-[3-(3-bromo-2-methyl-imidazo[1,2-a]pyrid...)
Affinity DataIC50: 380nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062886([3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-yloxy...)
Affinity DataIC50: 410nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062888(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 420nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062906(3-Bromo-2-methyl-8-(2,3,6-trichloro-benzyloxy)-imi...)
Affinity DataIC50: 490nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062908(Acetic acid {[3-(3-bromo-2-methyl-imidazo[1,2-a]py...)
Affinity DataIC50: 500nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062879(3-Bromo-8-(2,6-dichloro-3-methoxy-benzyloxy)-2-met...)
Affinity DataIC50: 540nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062907(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 580nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062876(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 580nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062903(2-Acetylamino-N-[3-(3-bromo-2-methyl-imidazo[1,2-a...)
Affinity DataIC50: 770nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062889(3-Acetylamino-N-[3-(3-bromo-2-methyl-imidazo[1,2-a...)
Affinity DataIC50: 810nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062881((3-Chloro-2-methyl-imidazo[1,2-a]pyridin-8-yl)-(2,...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062869([3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-yloxy...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062882(3-Bromo-8-(2-chloro-6-fluoro-benzyloxy)-2-methyl-i...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062885(3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-yloxym...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062892(2-(Acetyl-methyl-amino)-N-[3-(3-bromo-2-methyl-imi...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062862(3-Chloro-8-(2,6-dibromo-benzyloxy)-2-methyl-imidaz...)
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062873(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062870(3-Chloro-8-(2,6-difluoro-benzyloxy)-2-methyl-imida...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062894(N-[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-ylo...)
Affinity DataIC50: 2.10E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062866(8-(2,6-Dichloro-benzyloxy)-2-methyl-imidazo[1,2-a]...)
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062900([8-(2,6-Dichloro-benzyloxy)-2-methyl-imidazo[1,2-a...)
Affinity DataIC50: 7.50E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062902(8-(2,6-Dichloro-benzyloxy)-2-methyl-3-prop-2-ynylo...)
Affinity DataIC50: 7.60E+3nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062872(8-(2,6-Dichloro-benzyloxy)-2-ethyl-imidazo[1,2-a]p...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062877(8-(2,6-Dichloro-benzyloxy)-imidazo[1,2-a]pyridine ...)
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062904(1-Ethyl-5-methyl-2-[4-(2-methyl-quinolin-4-yloxyme...)
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062887(3-Bromo-8-(2,6-dichloro-phenoxymethyl)-2-methyl-im...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062861(3-Bromo-8-[(E)-2-(2,6-dichloro-phenyl)-vinyl]-2-me...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062895(N-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-yl)-N-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062875(3-Bromo-2-methyl-imidazo[1,2-a]pyridine-8-carboxyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062897(3-Bromo-2-methyl-imidazo[1,2-a]pyridine-8-carboxyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062874(8-(2,6-Dichloro-benzyloxy)-2-trifluoromethyl-imida...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062896(8-(2,6-Dichloro-benzyloxy)-2-methyl-imidazo[1,2-a]...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062880(2,6-Dichloro-N-(3-chloro-2-methyl-imidazo[1,2-a]py...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of specific binding of [3H]BK (0.06 nM) to bradykinin receptor B2 in guinea pig ileum membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed