Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 5130
LigandPNGBDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  0.870nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  1.06nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKi:  1.24nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  1.37nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  1.41nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  1.88nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  2.04nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  13.9nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM25878(Flunitrazepam | [3H]Rohypnol | 5-(2-fluorophenyl)-...)
Affinity DataKi:  14.9nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019213(5-(2-chlorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benz...)
Affinity DataKi:  18.6nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  24.5nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  28.3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  30.8nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50019213(5-(2-chlorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benz...)
Affinity DataKi:  33.4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  34.8nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  37.4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM25878(Flunitrazepam | [3H]Rohypnol | 5-(2-fluorophenyl)-...)
Affinity DataKi:  40.4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM23620(Dipyridamine | SMR000058382 | MLS000028420 | CHEMB...)
Affinity DataKi:  87.9nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM23620(Dipyridamine | SMR000058382 | MLS000028420 | CHEMB...)
Affinity DataKi:  162nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  187nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  193nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  616nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  622nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  644nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  767nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50244035(cid_105078 | Beta CCE | CHEMBL454606 | ethyl 9H-py...)
Affinity DataKi:  2.92E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM25878(Flunitrazepam | [3H]Rohypnol | 5-(2-fluorophenyl)-...)
Affinity DataKi:  3.14E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM25878(Flunitrazepam | [3H]Rohypnol | 5-(2-fluorophenyl)-...)
Affinity DataKi:  3.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  3.86E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019213(5-(2-chlorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benz...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019213(5-(2-chlorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benz...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed