Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50007286
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060785([D or LAgl (hydroxyacetic acid)4]acyline | CHEMBL2...)
Affinity DataIC50: 0.0560nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060807([L-3Pal3]acyline | CHEMBL216519)
Affinity DataIC50: 0.230nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060811([Ac-D or LAgl (Me,2-naphthoyl)1]acyline | CHEMBL41...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060776([D/LAgl (4-hydroxybenzoyl)5]acyline | CHEMBL262825)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060779([L or DAgl (hydroxyacetic acid)4]acyline | CHEMBL4...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060786([Ac-D2Nal1,D4Cpa2,D3Pal3,4Aph5(Ac),D4Aph6(Ac),ILys...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060775([L-Ala10]acyline | CHEMBL413752)
Affinity DataIC50: 0.380nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060778([D/LAgl (Me, 4-(acetylamino)benzoyl)5]acyline | CH...)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060794([D/LAgl10]acyline | CHEMBL2370593)
Affinity DataIC50: 0.480nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060795([D or LAgl (Me, isopropyl--Ala)8]acyline | CHEMBL2...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060806([D/LAgl (4-(acetylamino)benzoyl)5]acyline | CHEMBL...)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060791([D/LAgl (Me/isobutyryl)7]acyline | CHEMBL2370592)
Affinity DataIC50: 0.530nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060792([D or LAgl (formyl)10]acyline | CHEMBL407615)
Affinity DataIC50: 0.590nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060809([L or DAgl (formyl)10]acyline | CHEMBL267642)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060770([D or LAgl (formyl)4]acyline | CHEMBL407058)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060773([L or DAgl (nicotinoyl)3]acyline | CHEMBL262842)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060802([Ac-L-2Nal1]acyline | CHEMBL414558)
Affinity DataIC50: 0.640nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060774([D/LAgl (Me,formyl)10]acyline | CHEMBL2370594)
Affinity DataIC50: 0.670nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060787([D/LAgl (guanidinoacetyl)8]acyline | CHEMBL414469)
Affinity DataIC50: 0.740nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060801([D or LAgl (nicotinoyl)3]acyline | CHEMBL414468)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060805([L or LAgl (formyl)4]acyline | CHEMBL410798)
Affinity DataIC50: 0.840nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060808([Ac-L or DAgl (2-naphthoyl)1]acyline | CHEMBL43668...)
Affinity DataIC50: 0.880nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060789([D or LAgl (Me,formyl)4]acyline | CHEMBL262309)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060799([D/LAgl (Me)10]acyline | CHEMBL2370589)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060777([L or DAgl (Me,4-Cl-benzoyl)2]acyline | CHEMBL4299...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060803([L or DAgl (isonicotinoyl)3]acyline | CHEMBL436897)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060800([D/LAgl (Me,Ac)7]acyline | CHEMBL405736)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060797([L or DAgl (Me, 4-(acetylamino)benzoyl)6]acyline |...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060793([Dpr (isobutyryl)7]acyline | CHEMBL410799)
Affinity DataIC50: 2nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060804([D/LAgl (isobutyryl)7]acyline | CHEMBL269097)
Affinity DataIC50: 2nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060782([L or DAgl (Me, isopropyl--Ala)8]acyline | CHEMBL4...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060796([Ac-D or LAgl (2-naphthoyl)1]acyline | CHEMBL41345...)
Affinity DataIC50: 3nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060790(D/LAgl (Ac)7]acyline | CHEMBL444903)
Affinity DataIC50: 5nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060810([D or LAgl (Me, 4-(acetylamino)benzoyl)6]acyline |...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060781([L or DAgl (Me,formyl)4]acyline | CHEMBL263629)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060784([Ac-L or DAgl (Me,2-naphthoyl)1]acyline | CHEMBL26...)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060771([D or LAgl (Me,nicotinoyl)3]acyline | CHEMBL407193)
Affinity DataIC50: 36nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060798([D or LAgl (isonicotinoyl)3]acyline | CHEMBL439258)
Affinity DataIC50: 220nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50291968([D or LAgl (Me,4-Cl-benzoyl)2]acyline | CHEMBL2161...)
Affinity DataIC50: 280nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060780([L or DAgl (Apc)2]acyline | CHEMBL406211)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060788([D or LAgl (Pca)2]acyline | CHEMBL429381)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060772([L or DAgl (Pca)2]acyline | CHEMBL384385)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50060783([D or LAgL (Apc)2]acyline | CHEMBL263200)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed