Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50036549
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060064(2-[(R)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  2.5nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060071(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKd:  3.20nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060082(2-({2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-met...)
Affinity DataKd:  1.59E+3nMAssay Description:Antagonist activity against Opioid receptor mu 1 iin a guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060076(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKd:  1.00E+4nMAssay Description:Antagonist activity against Opioid receptor mu 1 iin a guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060065(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  0.126nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060082(2-({2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-met...)
Affinity DataKd:  0.251nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060068(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  1.59E+3nMAssay Description:Antagonist activity against Opioid receptor mu 1 iin a guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060075(2-({2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKd:  1.60nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060072(2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKd:  158nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060068(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  0.398nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060076(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKd:  2.5nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060065(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  501nMAssay Description:Antagonist activity against Opioid receptor mu 1 iin a guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.540nMAssay Description:Agonist activity for Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50059841(CHEMBL278789 | (S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-...)
Affinity DataIC50: 1.80nMAssay Description:Agonist activity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060076(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50454645(CHEMBL2370384)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060083(2-({2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060072(2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060075(2-({2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060071(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060064(2-[(R)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 in an in vitro guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060083(2-({2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  0.0755nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060068(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKi:  0.118nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060082(2-({2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-met...)
Affinity DataKi:  0.136nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060071(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  0.203nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060075(2-({2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  0.285nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50454645(CHEMBL2370384)
Affinity DataKi:  0.285nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060065(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKi:  0.310nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060076(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060073(2-[2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-(2S)-p...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060072(2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060064(2-[(R)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060081(2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  11nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060080(2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  13nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060079(2-[(S)-2-Dimethylamino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  44nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060066(2-[3-(4-Hydroxy-phenyl)-2-methylamino-propionyl]-1...)
Affinity DataKi:  75nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060084(2-({2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-met...)
Affinity DataKi:  106nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060077(2-({2-[(R)-2-Dimethylamino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  108nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi:  124nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060073(2-[2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-(2S)-p...)
Affinity DataKi:  277nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060071(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  379nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060065(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKi:  511nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060076(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  955nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060074(2-[3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyl-prop...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060081(2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  1.33E+3nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060083(2-({2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  1.52E+3nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060072(2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060068(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKi:  2.44E+3nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060080(2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  2.56E+3nMAssay Description:Binding affinity for Opioid receptor mu 1 by displacement of [3H]- DAGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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