Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50003461
Target5-hydroxytryptamine receptor 2C(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  5.50E+3nMAssay Description:Affinity pKi for 5-hydroxytryptamine 2C receptor was measured in rat cortex homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  5.62E+3nMAssay Description:Affinity pKi for Alpha-2 adrenergic receptor was measured in rat cortex homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  7.94E+3nMAssay Description:Affinity pKi for 5-hydroxytryptamine 2A receptor was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  9.33E+3nMAssay Description:Affinity pKi for 5-hydroxytryptamine 1A receptor was measured in rat cortex homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  1.00E+4nMAssay Description:Affinity pKi for 5-hydroxytryptamine 1D receptor was measured in calf caudate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  1.07E+4nMAssay Description:Affinity pKi for Dopamine receptor D2 was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  1.12E+4nMAssay Description:Affinity pKi for Alpha-1 adrenergic receptor was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  3.24E+4nMAssay Description:Affinity pKi for Dopamine receptor D1 was measured in rat cortex homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  4.57E+4nMAssay Description:Affinity pKi for Beta adrenergic receptor was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed