Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 5106
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85135(RS 57639)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85135(RS 57639)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85135(RS 57639)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50005836(4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50056404(BIMU 8 | CHEMBL59834 | 3-Isopropyl-2-oxo-2,3-dihyd...)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50056401(SDZ-205557 | SDZ 205557 | 2-diethylaminoethyl [2-m...)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50056401(SDZ-205557 | SDZ 205557 | 2-diethylaminoethyl [2-m...)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50056401(SDZ-205557 | SDZ 205557 | 2-diethylaminoethyl [2-m...)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82422(NSC_3035240 | CAS_109872-41-5 | RENZAPRIDE)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50056404(BIMU 8 | CHEMBL59834 | 3-Isopropyl-2-oxo-2,3-dihyd...)
Affinity DataKi:  50.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50007863(DAU 6285 | CHEMBL552854 | 6-Methoxy-2-oxo-2,3-dihy...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50005836(4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50007863(DAU 6285 | CHEMBL552854 | 6-Methoxy-2-oxo-2,3-dihy...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50056404(BIMU 8 | CHEMBL59834 | 3-Isopropyl-2-oxo-2,3-dihyd...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  126nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  126nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50007863(DAU 6285 | CHEMBL552854 | 6-Methoxy-2-oxo-2,3-dihy...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50005836(4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82422(NSC_3035240 | CAS_109872-41-5 | RENZAPRIDE)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82422(NSC_3035240 | CAS_109872-41-5 | RENZAPRIDE)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM81781(5-HT,omega-N-Me | 5-HT,a-Me)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  794nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  794nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  794nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  1.26E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  1.26E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM81781(5-HT,omega-N-Me | 5-HT,a-Me)
Affinity DataKi:  2.51E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataKi:  3.16E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM81781(5-HT,omega-N-Me | 5-HT,a-Me)
Affinity DataKi:  5.01E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataKi:  5.01E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed