Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50007030
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057114((2-Benzooxazol-6-yl-ethyl)-((R)-5-methoxy-1,2,3,4-...)
Affinity DataIC50: 5.25nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057102([2-(2-Methanesulfonyl-2,3-dihydro-1H-isoindol-5-yl...)
Affinity DataIC50: 5.81nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 6.43nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057099([2-(2,2-Dioxo-2,3-dihydro-1H-2lambda*6*-benzo[c]th...)
Affinity DataIC50: 6.67nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057101((2-Benzothiazol-6-yl-ethyl)-((R)-5-methoxy-1,2,3,4...)
Affinity DataIC50: 8.94nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057108(6-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50: 9.47nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057135([2-(1H-Benzoimidazol-5-yl)-ethyl]-((R)-5-methoxy-1...)
Affinity DataIC50: 11.3nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057124([2-(2,3-Dihydro-1H-isoindol-5-yl)-ethyl]-((R)-5-me...)
Affinity DataIC50: 11.6nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057098((2-Benzo[1,3]dioxol-5-yl-ethyl)-((R)-5-methoxy-1,2...)
Affinity DataIC50: 12.7nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057128(A-80426 | (2-Benzofuran-6-yl-ethyl)-((R)-5-methoxy...)
Affinity DataIC50: 13.1nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057113([2-(2,3-Dihydro-benzofuran-5-yl)-ethyl]-((R)-5-met...)
Affinity DataIC50: 14.6nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057110(5-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50: 16.3nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057104((2-Benzooxazol-5-yl-ethyl)-((R)-5-methoxy-1,2,3,4-...)
Affinity DataIC50: 16.7nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057142((2-Benzofuran-5-yl-ethyl)-((R)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50: 17.6nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057125([2-(2,3-Dihydro-benzofuran-6-yl)-ethyl]-((R)-5-met...)
Affinity DataIC50: 18.1nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057145(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 18.1nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057131(6-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50: 19.4nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057129((2-Indan-5-yl-ethyl)-((R)-5-methoxy-1,2,3,4-tetrah...)
Affinity DataIC50: 20.5nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057093((2-Benzo[1,3]dioxol-5-yl-ethyl)-(5-methoxy-1,2,3,4...)
Affinity DataIC50: 20.6nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057095(5-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50: 22.2nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057112([2-(2,3-Dihydro-benzo[b]thiophen-5-yl)-ethyl]-((R)...)
Affinity DataIC50: 24.3nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057126((2-Benzo[1,3]dioxol-5-yl-ethyl)-[(R)-1-(2,3,6,7,8,...)
Affinity DataIC50: 26.7nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057141([2-(2,3-Dihydro-1H-indol-5-yl)-ethyl]-((R)-5-metho...)
Affinity DataIC50: 31.8nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057111([2-(1,1-Dioxo-2,3-dihydro-1H-1lambda*6*-benzo[b]th...)
Affinity DataIC50: 33.7nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057092([2-(1-Methanesulfonyl-2,3-dihydro-1H-indol-5-yl)-e...)
Affinity DataIC50: 35nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057146([2-(2-Chloro-benzothiazol-6-yl)-ethyl]-((R)-5-meth...)
Affinity DataIC50: 38.2nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057147([2-(1-Methanesulfonyl-2,3-dihydro-1H-indol-6-yl)-e...)
Affinity DataIC50: 38.9nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057105(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 42.8nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057109(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 44.4nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057094(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 46.7nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057091([2-(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophen-5-yl)...)
Affinity DataIC50: 51nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057136((2-Benzo[b]thiophen-5-yl-ethyl)-((R)-5-methoxy-1,2...)
Affinity DataIC50: 52.8nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057097((2-Isoquinolin-7-yl-ethyl)-((R)-5-methoxy-1,2,3,4-...)
Affinity DataIC50: 53.9nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057123(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 59.8nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057134((2-Benzo[1,3]dioxol-5-yl-ethyl)-methyl-(6,7,8,9-te...)
Affinity DataIC50: 60.3nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057122(5-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50: 68.3nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057130([2-(2,3-Dihydro-1H-indol-6-yl)-ethyl]-((R)-5-metho...)
Affinity DataIC50: 79.1nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057107(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 86.7nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057139((2-Benzo[1,3]dioxol-5-yl-ethyl)-methyl-[(R)-1-(6,7...)
Affinity DataIC50: 101nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057138((2-Benzo[1,3]dioxol-5-yl-ethyl)-methyl-(5-methylsu...)
Affinity DataIC50: 117nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057143(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 132nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057127((2-Benzo[1,3]dioxol-5-yl-ethyl)-ethyl-((R)-5-metho...)
Affinity DataIC50: 158nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057132(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50: 183nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057103((2-Benzo[1,3]dioxol-5-yl-ethyl)-((R)-5-ethoxy-1,2,...)
Affinity DataIC50: 198nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057116([2-(1,3-Dihydro-isobenzofuran-5-yl)-ethyl]-((R)-5-...)
Affinity DataIC50: 229nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057133((2-Benzo[1,3]dioxol-5-yl-ethyl)-((R)-5-methoxy-1,2...)
Affinity DataIC50: 414nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057100((2-Benzo[1,3]dioxol-5-yl-ethyl)-[(3aS,6R)-1-(2,3,3...)
Affinity DataIC50: 436nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057106((2-Benzo[1,3]dioxol-5-yl-ethyl)-(6-methoxy-1,2,3,4...)
Affinity DataIC50: 469nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057140(N-(5-{[(2-Benzo[1,3]dioxol-5-yl-ethyl)-methyl-amin...)
Affinity DataIC50: 658nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057119((2-Benzo[1,3]dioxol-5-yl-ethyl)-((R)-5,6-dimethoxy...)
Affinity DataIC50: 757nMAssay Description:Inhibition of uptake of [3H]5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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