Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50006950
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50037078(2-(Phenyl)-isothiazolo[5,4-b]pyridin-3(2H)-one | c...)
Affinity DataIC50: 190nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056046(2-Pyridin-4-yl-isothiazolo[5,4-b]pyridin-3-one | C...)
Affinity DataIC50: 220nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50241343(H-168/68 | 5-methoxy-2-(2-(4-methoxy-3,5-dimethylp...)
Affinity DataIC50: 370nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056043(2-(2,4-Diethoxy-phenylmethanesulfinyl)-N-pyridin-4...)
Affinity DataIC50: 400nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056045(2-(2-Ethoxy-4-methoxy-phenylmethanesulfinyl)-N-pyr...)
Affinity DataIC50: 450nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056041(2-(2,4-Dimethoxy-6-methyl-phenylmethanesulfinyl)-N...)
Affinity DataIC50: 460nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056049(2-Isobutyl-isothiazolo[5,4-b]pyridin-3-one | CHEMB...)
Affinity DataIC50: 530nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056056(2-(2,4-Dimethoxy-phenylmethanesulfinyl)-N-pyridin-...)
Affinity DataIC50: 590nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056042(N-Pyridin-4-yl-2-(2,4,6-trimethoxy-phenylmethanesu...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056050(2-(Di-p-tolyl-methanesulfinyl)-N-pyridin-4-yl-nico...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056051(2-[2-(2-Fluoro-ethoxy)-4-methoxy-phenylmethanesulf...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056047(2-(5-Bromo-2,4-dimethoxy-phenylmethanesulfinyl)-N-...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056042(N-Pyridin-4-yl-2-(2,4,6-trimethoxy-phenylmethanesu...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056044(2-(2,4-Dimethoxy-3-methyl-phenylmethanesulfinyl)-N...)
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056052(2-(2,6-Dimethoxy-phenylmethanesulfinyl)-N-pyridin-...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056054(2-[2-(2-Hydroxy-ethoxy)-4-methoxy-phenylmethanesul...)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of [14C]aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056043(2-(2,4-Diethoxy-phenylmethanesulfinyl)-N-pyridin-4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056056(2-(2,4-Dimethoxy-phenylmethanesulfinyl)-N-pyridin-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056041(2-(2,4-Dimethoxy-6-methyl-phenylmethanesulfinyl)-N...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056052(2-(2,6-Dimethoxy-phenylmethanesulfinyl)-N-pyridin-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056045(2-(2-Ethoxy-4-methoxy-phenylmethanesulfinyl)-N-pyr...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056051(2-[2-(2-Fluoro-ethoxy)-4-methoxy-phenylmethanesulf...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056048(N-Pyridin-4-yl-2-(2,4,5-trimethoxy-phenylmethanesu...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056044(2-(2,4-Dimethoxy-3-methyl-phenylmethanesulfinyl)-N...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed