Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50042212
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.320nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.630nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50329178((S)-3-(3-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl...)
Affinity DataIC50: 10nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50422183(CHEMBL358778)
Affinity DataIC50: 10nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50422182(CHEMBL356408)
Affinity DataIC50: 16nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50072427(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataIC50: 25nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50072427(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataIC50: 50nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50329178((S)-3-(3-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl...)
Affinity DataIC50: 126nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50422183(CHEMBL358778)
Affinity DataIC50: 200nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM50422182(CHEMBL356408)
Affinity DataIC50: 316nMAssay Description:Compound was tested in vitro for its ability to displace [125I]Bolton-Hunter CCK-8 from membrane preparation isolated from CHO-KI cells stably transf...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed