Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50042078
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420244(CHEMBL1628111)
Affinity DataKi:  1.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50366524(Estrone Sulphate | ESTRONE | ESTROPIPATE | Estrone...)
Affinity DataKi:  1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420245(CHEMBL1614647)
Affinity DataKi:  1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420242(CHEMBL2075012)
Affinity DataKi:  1.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420249(CHEMBL2074598)
Affinity DataKi:  2.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420248(CHEMBL2074651)
Affinity DataKi:  3.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataKi:  4.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50170653(11beta,21-dihydroxypregn-4-ene-3,20-dione | cortic...)
Affinity DataKi:  5.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM8885(Testosterone, 1 | (1S,2R,10R,11S,14S,15S)-14-hydro...)
Affinity DataKi:  5.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420246(CHEMBL2074591)
Affinity DataKi:  9.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50410506(ESTRIOL)
Affinity DataKi:  9.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM17639((1S,2S,5R,7S,10R,11S,15S)-5-hydroxy-2,15-dimethylt...)
Affinity DataKi:  1.06E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM17289(folliculin | (1S,10R,11S,15S)-5-hydroxy-15-methylt...)
Affinity DataKi:  1.57E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420243(CHEMBL2074705)
Affinity DataKi:  7.62E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1A1(Rat)
Albert Einstein College of Medicine

Curated by ChEMBL
LigandPNGBDBM50420247(CHEMBL2074716)
Affinity DataKi: >2.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed