Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50036439
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50052440(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  0.0540nMAssay Description:Inhibitory constant for RTX binding to rat spinal cordMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50052440(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  0.120nMAssay Description:Inhibitory constant for RTX binding to porcine spinal cordMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50052440(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  0.450nMAssay Description:Inhibitory constant for RTX binding to human spinal cordMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50052437(4-Azido-benzoic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9a...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052439((4-Azido-phenyl)-acetic acid (1aR,1bS,4aR,7aS,7bS,...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052443(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052445(Benzoic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-9a-ac...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052441(Cyclohexyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052440(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]RTX binding from Vanilloid receptor of rat dorsal Root Ganglion (DRG) membranesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM20284(N-[2-(4-chlorophenyl)ethyl]-7,8-dihydroxy-2,3,4,5-...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50052447(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bR,8S,9aS)-4a...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052446(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50052440(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]- RTX binding to vanilloid receptor of rat urinary bladderMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50052440(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of [3H]- RTX binding to Vanilloid receptors from pig spinal cordMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052448(Cyclohexanecarboxylic acid (1aR,1bS,4aR,7aS,7bS,8R...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052440(Phenyl-acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibition of [3H]- RTX binding to Vanilloid receptors from human spinal cordMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052438(Phenyl-acetic acid (1aR,1bS,4aR,5S,7aS,7bS,8R,9R,9...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50052444((4-Hydroxy-3-methoxy-phenyl)-acetic acid (1aR,1bS,...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed