Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50036425
TargetAdenylate cyclase type 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051588(His-Ser-Gln-thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataEC50:  8nMAssay Description:Ability of the Compound to activate Adenylate cyclase activity was measured by the conversion of [alpha-32P]ATP to 3'5'-cyclic AMPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051588(His-Ser-Gln-thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051586([des-His1,Tyr5,Glu9,D-Tyr10]glucagon-NH2 | CHEMBL4...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50407844(CHEMBL2115191)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50454201(CHEMBL3037804)
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50407842(CHEMBL2114176)
Affinity DataIC50: 34.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051585([des-His1,Tyr5,Glu9,(2S,3R)-beta-MePhe10]glucagon-...)
Affinity DataIC50: 74nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)
Affinity DataIC50: 170nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)
Affinity DataIC50: 180nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50407843(CHEMBL2114177)
Affinity DataIC50: 395nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50407841(CHEMBL2115192)
Affinity DataIC50: 510nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed