Compile Data Set for Download or QSAR
Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 50036154
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045224(Ac-D-Dip-Leu-Phe-Ile-Ile-Trp | CHEMBL387200)
Affinity DataEC50:  580nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045234(Ac-D-Dip-Leu-Asp-Ile-Ile-Tyr | CHEMBL313344)
Affinity DataEC50:  2.70E+3nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045246(Ac-D-Dip-Orn-Asp-Ile-Ile-Trp | CHEMBL2370066)
Affinity DataEC50:  13nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045249(Ac-D-Dip-Leu-Asp-Ile-Val-Trp | CHEMBL86703)
Affinity DataEC50:  6.00E+3nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045246(Ac-D-Dip-Orn-Asp-Ile-Ile-Trp | CHEMBL2370066)
Affinity DataEC50:  13nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045224(Ac-D-Dip-Leu-Phe-Ile-Ile-Trp | CHEMBL387200)
Affinity DataEC50:  60nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045256(D-Dip-Leu-Asp-Ile-Ile-Trp | CHEMBL2370067)
Affinity DataEC50:  1.90E+3nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045256(D-Dip-Leu-Asp-Ile-Ile-Trp | CHEMBL2370067)
Affinity DataEC50:  1.90E+3nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045234(Ac-D-Dip-Leu-Asp-Ile-Ile-Tyr | CHEMBL313344)
Affinity DataEC50:  6.10E+3nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045264(Ac-D-Dip-Leu-Asp-Val-Ile-Trp | CHEMBL315841)
Affinity DataEC50:  17nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045249(Ac-D-Dip-Leu-Asp-Ile-Val-Trp | CHEMBL86703)
Affinity DataEC50:  6.00E+3nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045263(Ac-D-Dip-Glu-Asp-Ile-Ile-Trp | CHEMBL407269)
Affinity DataEC50:  52nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045263(Ac-D-Dip-Glu-Asp-Ile-Ile-Trp | CHEMBL407269)
Affinity DataEC50:  25nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045264(Ac-D-Dip-Leu-Asp-Val-Ile-Trp | CHEMBL315841)
Affinity DataEC50:  50nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045239(Ac-D-Dip-Leu-Asp-Ile-Ile-Trp | Ac-D-Dip-Leu-Asp-Il...)
Affinity DataIC50: 25nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045240(Ac-D-Phe-Leu-Phe-Ile-Ile-Trp | (S)-2-[(S)-2-((2S,5...)
Affinity DataIC50: 36nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368647(CHEMBL1788127)
Affinity DataIC50: 40nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 60nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 60nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368647(CHEMBL1788127)
Affinity DataIC50: 60nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045239(Ac-D-Dip-Leu-Asp-Ile-Ile-Trp | Ac-D-Dip-Leu-Asp-Il...)
Affinity DataIC50: 70nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368647(CHEMBL1788127)
Affinity DataIC50: 70nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045230(Ac-D-Trp-Leu-Asp-Ile-Ile-Trp | CHEMBL313382)
Affinity DataIC50: 130nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045239(Ac-D-Dip-Leu-Asp-Ile-Ile-Trp | Ac-D-Dip-Leu-Asp-Il...)
Affinity DataIC50: 140nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045257(Ac-D-Phe-Leu-Asp-Ile-Ile-Tyr | CHEMBL89736)
Affinity DataIC50: 150nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 200nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 200nMAssay Description:Binding affinity against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001219(CHEMBL85341 | 3-{2-[2-Acetylamino-3-(4-hydroxy-phe...)
Affinity DataIC50: 250nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045262(Ac-D-Phe-Ala-Asp-Ile-Ile-Trp | CHEMBL406279)
Affinity DataIC50: 290nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 330nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045240(Ac-D-Phe-Leu-Phe-Ile-Ile-Trp | (S)-2-[(S)-2-((2S,5...)
Affinity DataIC50: 380nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001219(CHEMBL85341 | 3-{2-[2-Acetylamino-3-(4-hydroxy-phe...)
Affinity DataIC50: 400nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045262(Ac-D-Phe-Ala-Asp-Ile-Ile-Trp | CHEMBL406279)
Affinity DataIC50: 420nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045262(Ac-D-Phe-Ala-Asp-Ile-Ile-Trp | CHEMBL406279)
Affinity DataIC50: 420nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045230(Ac-D-Trp-Leu-Asp-Ile-Ile-Trp | CHEMBL313382)
Affinity DataIC50: 450nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045237(Ac-D-Phe-Leu-Asp-Ala-Ile-Trp | CHEMBL87243)
Affinity DataIC50: 450nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045227(Ac-D-Phe-Orn-Asp-Ile-Ile-Trp | (S)-3-[2-((R)-2-Ace...)
Affinity DataIC50: 680nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045243(Ac-D-Phe-Glu-Asp-Ile-Trp | CHEMBL313056)
Affinity DataIC50: 740nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 740nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045243(Ac-D-Phe-Glu-Asp-Ile-Trp | CHEMBL313056)
Affinity DataIC50: 840nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045243(Ac-D-Phe-Glu-Asp-Ile-Trp | CHEMBL313056)
Affinity DataIC50: 930nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001221(CHEMBL315047 | 3-[2-(2-Acetylamino-3-naphthalen-2-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001221(CHEMBL315047 | 3-[2-(2-Acetylamino-3-naphthalen-2-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045240(Ac-D-Phe-Leu-Phe-Ile-Ile-Trp | (S)-2-[(S)-2-((2S,5...)
Affinity DataIC50: 1.40E+3nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045237(Ac-D-Phe-Leu-Asp-Ala-Ile-Trp | CHEMBL87243)
Affinity DataIC50: 1.61E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045230(Ac-D-Trp-Leu-Asp-Ile-Ile-Trp | CHEMBL313382)
Affinity DataIC50: 1.80E+3nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 1.80E+3nMAssay Description:Effective concentration against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001221(CHEMBL315047 | 3-[2-(2-Acetylamino-3-naphthalen-2-...)
Affinity DataIC50: 1.90E+3nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 2.00E+3nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045251(Ac-D-Phe-Asp-Ile-Ile-Trp | 3-((R)-2-Acetylamino-3-...)
Affinity DataIC50: 2.15E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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