Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50036276
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044039((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044033((S)-3-[(S)-2-((S)-2-Benzoylamino-3-1H-indol-3-yl-p...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044042((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[2...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044028((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044038((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044044((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044032((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044037((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044031((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040523((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044025((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044043((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044022((S)-3-[(S)-2-[2-Acetylamino-3-(1H-indol-3-yl)-prop...)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044024((S)-3-[(S)-2-[2-((S)-3-tert-Butyl-ureido)-3-(1H-in...)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044040((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044036((S)-3-[(S)-2-[(S)-2-Benzyloxycarbonylamino-3-(1H-i...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044023((S)-3-[(S)-2-[(S)-2-(Adamantan-2-yloxycarbonylamin...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044029((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044030((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 13nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044034((S)-3-[(S)-2-[(S)-2-(Adamantan-1-yloxycarbonylamin...)
Affinity DataIC50: 17nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044026((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 18nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044027((S)-3-[(S)-2-[(S)-2-(2-Adamantan-1-yl-acetylamino)...)
Affinity DataIC50: 19nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044041(methylsulfonyl-Trp-Lys(Tac)-Asp-N(Me)-Phe-NH2 | CH...)
Affinity DataIC50: 41nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044038((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 42nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044035(N-{(S)-1-[(S)-1-{1-[(S)-((S)-1-Carbamoyl-2-phenyl-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044035(N-{(S)-1-[(S)-1-{1-[(S)-((S)-1-Carbamoyl-2-phenyl-...)
Affinity DataIC50: 2.50E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044031((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 3.00E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044024((S)-3-[(S)-2-[2-((S)-3-tert-Butyl-ureido)-3-(1H-in...)
Affinity DataIC50: 3.50E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044028((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 4.50E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044033((S)-3-[(S)-2-((S)-2-Benzoylamino-3-1H-indol-3-yl-p...)
Affinity DataIC50: 4.60E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040523((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 4.70E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044039((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 4.70E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044036((S)-3-[(S)-2-[(S)-2-Benzyloxycarbonylamino-3-(1H-i...)
Affinity DataIC50: 4.80E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044040((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 4.80E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044025((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 5.20E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044042((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[2...)
Affinity DataIC50: 5.20E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044044((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 5.70E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044037((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 6.10E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044032((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 6.10E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044022((S)-3-[(S)-2-[2-Acetylamino-3-(1H-indol-3-yl)-prop...)
Affinity DataIC50: 6.40E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044030((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 6.40E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044043((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 6.50E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044023((S)-3-[(S)-2-[(S)-2-(Adamantan-2-yloxycarbonylamin...)
Affinity DataIC50: 7.40E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50044026((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 7.60E+3nMAssay Description:Concentration required to inhibit 50% of specific binding to Cholecystokinin type B receptor in guinea pig cortex using [125I]Bolton-Hunter CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed