Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50036308
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  0.00720nMAssay Description:Tested for binding activity against delta1 opioid receptor using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040487(17-(cyclopropylmethyl)4,5-alpha-epoxy-3,14-dihydro...)
Affinity DataKi:  0.0470nMAssay Description:Tested for binding activity against delta opioid receptor using [3H]naltridole ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  0.100nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  0.120nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  0.190nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  0.600nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  0.830nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  0.860nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040487(17-(cyclopropylmethyl)4,5-alpha-epoxy-3,14-dihydro...)
Affinity DataKi:  1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  1.5nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  1.80nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  1.90nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  2.20nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  2.20nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  4.5nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  5.20nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  5.90nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040484(14-anilino-4-cyclopropylmethyl-(13R,14R,17S)-12-ox...)
Affinity DataKi:  7.80nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  10nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040485(15-benzyl-4-cyclopropylmethyl-10,17-dihydroxy-(1S,...)
Affinity DataKi:  13nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040487(17-(cyclopropylmethyl)4,5-alpha-epoxy-3,14-dihydro...)
Affinity DataKi:  13nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  14nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  14nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  15nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  25nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040483(4-cyclopropylmethyl-10,17-dihydroxy-15-phenyl-(1S,...)
Affinity DataKi:  25nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056628(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-phenyl-(...)
Affinity DataKi:  66nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50040482(17-(cyclopropylmethyl)-6,7-didehydro-4,5-alpha-epo...)
Affinity DataKi:  121nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed