Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50005716
TargetKappa-type opioid receptor(Guinea pig)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  0.150nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]bremazocineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  0.190nMAssay Description:Compound was tested for binding affinity towards mu-opioid receptor in rat forebrain membrane using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  3.90nMAssay Description:Compound was tested for binding affinity towards delta-opioid receptor in rat forebrain membrane using [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040187(Tyr-Aib-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  10nMAssay Description:Compound was tested for binding affinity towards mu-opioid receptor in rat forebrain membrane using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((trans)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-...)
Affinity DataKi:  13nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]bremazocineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((trans)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-...)
Affinity DataKi:  13nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]bremazocineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040187(Tyr-Aib-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  50nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]bremazocineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((trans)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-...)
Affinity DataKi:  117nMAssay Description:Compound was tested for binding affinity towards delta-opioid receptor in rat forebrain membrane using [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((trans)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-...)
Affinity DataKi:  275nMAssay Description:Compound was tested for binding affinity towards mu-opioid receptor in rat forebrain membrane using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((trans)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-...)
Affinity DataKi:  1.37E+3nMAssay Description:Compound was tested for binding affinity towards delta-opioid receptor in rat forebrain membrane using [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed