Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50005709
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040108(11-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethylsulfa...)
Affinity DataKi:  6.90nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002084(CHEMBL538750 | CHEMBL336317 | 11-(2-Dimethylamino-...)
Affinity DataKi:  9nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040114({11-[2-(4-Benzyl-piperidin-1-yl)-ethylsulfanyl]-6,...)
Affinity DataKi:  10nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002088(CHEMBL302005 | [11-(2-Dimethylamino-ethylidene)-6,...)
Affinity DataKi:  11nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040109(3-{11-[2-(4-Benzyl-piperidin-1-yl)-ethylsulfanyl]-...)
Affinity DataKi:  12nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040112(11-[2-(4-Benzyl-piperazin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  14nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50175516({11-[2-(4-Benzyl-piperidin-1-yl)-eth-(E)-ylidene]-...)
Affinity DataKi:  15nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040110(2-{11-[2-(4-Benzyl-piperidin-1-yl)-ethylsulfanyl]-...)
Affinity DataKi:  17nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040111({11-[2-(4-Benzyl-piperidin-1-yl)-ethylidene]-6,11-...)
Affinity DataKi:  20nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040121(11-[2-(4-Phenyl-piperidin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  20nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040113(11-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethylsu...)
Affinity DataKi:  41nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040116(11-(2-Morpholin-4-yl-ethylsulfanyl)-6,11-dihydro-d...)
Affinity DataKi:  42nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040119(11-[2-(4-Phenyl-piperazin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  47nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040117(11-{2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-pi...)
Affinity DataKi:  500nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040115(Sodium; 11-[2-(4-benzyl-piperidin-1-yl)-ethylsulfa...)
Affinity DataKi:  740nMAssay Description:Inhibition of the specific binding of [3H]pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed