Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50036287
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 1.30E+3nMAssay Description:Tested for competitive inhibition of endoplasmic reticulum alpha-glucosidase II.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50292389(3-epifagomine | 3-epi-fagomine | CHEMBL456583)
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for competitive inhibition of bovine liver beta-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLactase/phlorizin hydrolase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50292389(3-epifagomine | 3-epi-fagomine | CHEMBL456583)
Affinity DataIC50: 1.90E+3nMAssay Description:Tested for competitive inhibition of rat intestinal lactaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50292389(3-epifagomine | 3-epi-fagomine | CHEMBL456583)
Affinity DataIC50: 3.10E+3nMAssay Description:Concentration that causes 50% inhibition of mammalian cytosolic beta-galactosidase was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 3.30E+3nMAssay Description:Concentration that causes 50% inhibition of mammalian cytosolic beta-galactosidase was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 3.60E+3nMAssay Description:Concentration that causes 50% inhibition of mammalian lactase beta-galactosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50292389(3-epifagomine | 3-epi-fagomine | CHEMBL456583)
Affinity DataIC50: 4.00E+3nMAssay Description:Concentration that causes 50% inhibition of mammalian lactase beta-galactosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrehalase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 4.80E+3nMAssay Description:Concentration that causes 50% inhibition of mammalian trehalase was determined in porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase C(Mouse)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 5.80E+3nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (isomaltase) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase C(Mouse)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50292389(3-epifagomine | 3-epi-fagomine | CHEMBL456583)
Affinity DataIC50: 6.40E+3nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (isomaltase) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50240725((2R,3R,4R)-2-Hydroxymethyl-piperidine-3,4-diol | F...)
Affinity DataIC50: 1.50E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian lactase beta-galactosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50403869(CHEMBL2115197)
Affinity DataIC50: 1.70E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian lactase beta-galactosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase C(Mouse)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50403869(CHEMBL2115197)
Affinity DataIC50: 1.70E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (isomaltase) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of mammalian alpha-glucosidase (lysosomal) was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of mammalian alpha-glucosidase (lysosomal) was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrehalase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 2.50E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian trehalase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.50E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-mannosidase (Golgi I) was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.50E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (lysosomal) was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLactase/phlorizin hydrolase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.60E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian lactase beta-galactosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTissue alpha-L-fucosidase(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.60E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-L-fucosidase was determined in bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.70E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian beta-galactosidase (lactase ) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 3.00E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian lactase beta-galactosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 3.40E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian cellobiase beta-glucosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase C(Mouse)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 3.40E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (isomaltase) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase C(Mouse)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 3.40E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (isomaltase) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50240725((2R,3R,4R)-2-Hydroxymethyl-piperidine-3,4-diol | F...)
Affinity DataIC50: 3.80E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian cytosolic beta-galactosidase was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrehalase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 4.10E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian trehalase was determined in porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrehalase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 4.20E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian trehalase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 4.60E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-mannosidase (golgi II) was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 5.30E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-mannosidase (golgi I) was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 5.50E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (maltase) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 8.40E+4nMAssay Description:Concentration that causes 50% inhibition of soluble mammalian alpha-mannosidase in rat liver; NI is less than 50 % inhibition at 1000 uMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 8.40E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-mannosidase was determined in rat epididymisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of mammalian alpha-glucosidase (lysosomal) was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase C(Mouse)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 9.10E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (isomaltase) was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 9.20E+4nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (lysosomal) was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 1.00E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-glucosidase (lysosomal) was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50292389(3-epifagomine | 3-epi-fagomine | CHEMBL456583)
Affinity DataIC50: 1.00E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian cellobiase beta-glucosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 1.10E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-mannosidase (lysosomal) was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTissue alpha-L-fucosidase(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50240725((2R,3R,4R)-2-Hydroxymethyl-piperidine-3,4-diol | F...)
Affinity DataIC50: 1.40E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-L-fucosidase was determined in bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal alpha-glucosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of mammalian alpha-glucosidase (lysosomal) was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrehalase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 2.00E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian trehalase was determined in porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 2.10E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian alpha-mannosidase was determined in rat epididymisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50403869(CHEMBL2115197)
Affinity DataIC50: 2.30E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian cellobiase beta-glucosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLactase/phlorizin hydrolase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50407255(CHEMBL2114189)
Affinity DataIC50: 2.60E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian lactase beta-galactosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Bovine)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 3.00E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian cytosolic beta-galactosidase was determined in bovine liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeutral alpha-glucosidase AB(Human)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 3.20E+5nMAssay Description:Concentration that causes 50% inhibition of soluble mammalian alpha-mannosidase in rat liver. NI is less than 50 % inhibition at 1000 micro MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrehalase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataIC50: 3.60E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian trehalase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase(Rat)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 3.90E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian lysosomal beta-galactosidase was determined in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50: 4.60E+5nMAssay Description:Concentration that causes 50% inhibition of mammalian cellobiase beta-glucosidase was determined in rat intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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