Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50005357
Affinity DataKi: 1.5nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 was determined by measuring its ability to displace [3H]-AF-DX 384 from rat he...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 was determined by measuring its ability to displace [3H]-AF-DX 384 from rat he...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 was determined by measuring its ability to displace [3H]-AF-DX 384 from rat he...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 was determined by measuring its ability to displace [3H]pirenzepine from bovin...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 was determined by measuring its ability to displace [3H]-AF-DX 384 from rat he...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 was determined by measuring its ability to displace [3H]-AF-DX 384 from rat he...More data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 was determined by measuring its ability to displace [3H]pirenzepine from bovin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
National Institutes of Health
Curated by ChEMBL
National Institutes of Health
Curated by ChEMBL
Affinity DataKi: 18.6nMAssay Description:In vitro binding affinity towards Sigma receptor type 1 was determined by measuring its ability to displace [3H](+)-pentazocine from guinea pig brain...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
National Institutes of Health
Curated by ChEMBL
National Institutes of Health
Curated by ChEMBL
Affinity DataKi: 21.7nMAssay Description:In vitro binding affinity towards Sigma receptor type 1 was determined by measuring its ability to displace [3H](+)-pentazocine from guinea pig brain...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 was determined by measuring its ability to displace [3H]pirenzepine from bovin...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 was determined by measuring its ability to displace [3H]pirenzepine from bovin...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 was determined by measuring its ability to displace [3H]pirenzepine from bovin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
National Institutes of Health
Curated by ChEMBL
National Institutes of Health
Curated by ChEMBL
Affinity DataKi: 62.1nMAssay Description:In vitro binding affinity towards Sigma receptor type 1 was determined by measuring its ability to displace [3H](+)-pentazocine from guinea pig brain...More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- Scopolamine...More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- Scopolamine...More data for this Ligand-Target Pair
Affinity DataKi: 163nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- Scopolamine...More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:In vitro binding affinity towards Sigma receptor type 2 was determined by measuring its ability to displace [3H]1,3-di-o-tolylguanidine from rat live...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- Scopolamine...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- Scopolamine...More data for this Ligand-Target Pair
