Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 4880
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033312(Urapidil-5-methyl | CHEMBL539806 | Benzyl-(6-chlor...)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033312(Urapidil-5-methyl | CHEMBL539806 | Benzyl-(6-chlor...)
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM82424(CAS_1236 | NSC_1236 | Niguldipine(+))
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM82424(CAS_1236 | NSC_1236 | Niguldipine(+))
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Bovine)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033312(Urapidil-5-methyl | CHEMBL539806 | Benzyl-(6-chlor...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033312(Urapidil-5-methyl | CHEMBL539806 | Benzyl-(6-chlor...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  126nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033312(Urapidil-5-methyl | CHEMBL539806 | Benzyl-(6-chlor...)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM84342(EPINEPHRINE | 4-[1-hydroxy-2-(methylamino)ethyl]be...)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM50033312(Urapidil-5-methyl | CHEMBL539806 | Benzyl-(6-chlor...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Rat)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM82424(CAS_1236 | NSC_1236 | Niguldipine(+))
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1B adrenergic receptor(Hamster)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM82424(CAS_1236 | NSC_1236 | Niguldipine(+))
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM82424(CAS_1236 | NSC_1236 | Niguldipine(+))
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  794nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Human)
Duke University

Curated by PDSP Ki Database
LigandPNGBDBM82424(CAS_1236 | NSC_1236 | Niguldipine(+))
Affinity DataKi:  794nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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