Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50005207
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034281(Bicyclo[2.2.1]heptane-2-carboxylic acid {2-[4-(2-m...)
Affinity DataKi:  0.120nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034308(Bicyclo[2.2.1]heptane-2-carboxylic acid {4-[4-(2-m...)
Affinity DataKi:  0.230nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034292(Octahydro-pentalene-2-carboxylic acid {2-[4-(2-met...)
Affinity DataKi:  0.240nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034300(Bicyclo[2.2.1]hept-5-ene-2-carboxylic acid {2-[4-(...)
Affinity DataKi:  0.270nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034303(Bicyclo[2.2.1]hept-5-ene-2-carboxylic acid {4-[4-(...)
Affinity DataKi:  0.380nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034302(Octahydro-pentalene-2-carboxylic acid {4-[4-(2-met...)
Affinity DataKi:  0.630nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034296(1-Methyl-1H-pyrrole-2-carboxylic acid {4-[4-(2-met...)
Affinity DataKi:  0.740nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  1.18nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034288(1-Methyl-1H-pyrrole-2-carboxylic acid {2-[4-(2-met...)
Affinity DataKi:  1.19nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  1.26nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034309(3-Methyl-thiophene-2-carboxylic acid {4-[4-(2-meth...)
Affinity DataKi:  1.53nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034286(Cyclopentanecarboxylic acid {4-[4-(2-methoxy-pheny...)
Affinity DataKi:  1.88nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034282(Thiophene-3-carboxylic acid {4-[4-(2-methoxy-pheny...)
Affinity DataKi:  2.20nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034304(5-Methyl-thiophene-2-carboxylic acid {2-[4-(2-meth...)
Affinity DataKi:  2.29nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034284(Thiophene-2-carboxylic acid {4-[4-(2-methoxy-pheny...)
Affinity DataKi:  2.34nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034298(3-Methyl-thiophene-2-carboxylic acid {2-[4-(2-meth...)
Affinity DataKi:  3.09nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034301(3-Chloro-thiophene-2-carboxylic acid {4-[4-(2-meth...)
Affinity DataKi:  3.34nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034297(5-Methyl-thiophene-2-carboxylic acid {4-[4-(2-meth...)
Affinity DataKi:  3.80nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034295(Cyclopentanecarboxylic acid {2-[4-(2-methoxy-pheny...)
Affinity DataKi:  4.68nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034299(Thiophene-3-carboxylic acid {2-[4-(2-methoxy-pheny...)
Affinity DataKi:  6.83nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034290(Octahydro-pentalene-2-carboxylic acid {3-[4-(2-met...)
Affinity DataKi:  11.6nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034306(1H-Pyrrole-2-carboxylic acid {4-[4-(2-methoxy-phen...)
Affinity DataKi:  12.5nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  15.4nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034291(N-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  17.5nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034285(1H-Pyrrole-2-carboxylic acid {2-[4-(2-methoxy-phen...)
Affinity DataKi:  20.3nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034307(N-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  25.2nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034294(3-Methoxy-thiophene-2-carboxylic acid {4-[4-(2-met...)
Affinity DataKi:  32.1nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034293(N-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-...)
Affinity DataKi:  32.3nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034289(Furan-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-p...)
Affinity DataKi:  55.7nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034287(1H-Pyrrole-2-carboxylic acid {3-[4-(2-methoxy-phen...)
Affinity DataKi:  201nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034305(N-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataKi:  321nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Faes

Curated by ChEMBL
LigandPNGBDBM50034283(N-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-...)
Affinity DataKi:  362nMAssay Description:In vitro ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed