Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50036355
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033213(7,8-Dichloro-1-methyl-4-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033211(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033212(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033223(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.600nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033214(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.700nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033206(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.900nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033207(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 1.90nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033217(7,8-Dichloro-2-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 4nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004633(4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-imidaz...)
Affinity DataIC50: 4.30nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033218(1-Methyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50: 4.90nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033224(4-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50: 5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033215(2-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50: 15nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033219(2-Methyl-1-[4-(5-phenyl-[1,3,4]oxadiazol-2-yl)-phe...)
Affinity DataIC50: 44nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033226(1-(4-Iodo-phenyl)-2-methyl-1H-imidazo[4,5-c]pyridi...)
Affinity DataIC50: 67nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50038755(6-(2-chlorophenyl)-1-methyl-8,9-dihydro-4H,7H-cycl...)
Affinity DataIC50: 73nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033221(5-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50: 190nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033225(4-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50: 200nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033209(1-[4-(1H-Benzoimidazol-2-yl)-phenyl]-2-methyl-1H-i...)
Affinity DataIC50: 350nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033216(3-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50: 600nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033208(2-Methyl-1-phenyl-1H-imidazo[4,5-c]pyridine | CHEM...)
Affinity DataIC50: 840nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033222(7-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033220(5-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed