Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50003414
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470598(CHEMBL126050)
Affinity DataKi:  1nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470604(CHEMBL338825)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470590(CHEMBL341357)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470583(CHEMBL125696)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470596(CHEMBL125310)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  2.5nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470587(CHEMBL124648)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470605(CHEMBL122169)
Affinity DataKi:  4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470603(CHEMBL124013)
Affinity DataKi:  4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470582(CHEMBL126043)
Affinity DataKi:  5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470595(CHEMBL122019)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470599(CHEMBL330766)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  7.90nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470592(CHEMBL339311)
Affinity DataKi:  7.90nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470597(CHEMBL330826)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470606(CHEMBL446099)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470581(CHEMBL341008)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470584(CHEMBL125001)
Affinity DataKi:  13nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470585(CHEMBL415518)
Affinity DataKi:  16nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470608(CHEMBL338030)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470607(CHEMBL124624)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470601(CHEMBL123731)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470589(CHEMBL331011)
Affinity DataKi:  79nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470600(CHEMBL435619)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470602(CHEMBL340747)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470594(CHEMBL340405)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470586(CHEMBL435610)
Affinity DataKi:  126nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470593(CHEMBL126158)
Affinity DataKi:  200nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470588(CHEMBL340548)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  7.94E+3nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from rabbit cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi: <1.00E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  7.94E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 3 from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed