Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50035447
LigandPNGBDBM50029150(CHEMBL276520 | 3-(2-Piperidin-4-yl-ethyl)-1H-indol...)
Affinity DataIC50: 10nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029145(3-(2-Piperidin-4-yl-ethyl)-1H-indol-5-ol; fumarate)
Affinity DataIC50: 20nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM77970(CLOMIPRAMINE HYDROCHLORIDE | CHLORIMIPRAMINE | 3-(...)
Affinity DataIC50: 20nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029150(CHEMBL276520 | 3-(2-Piperidin-4-yl-ethyl)-1H-indol...)
Affinity DataIC50: 30nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029140(3-(3-Piperidin-4-yl-propyl)-1H-indole | CHEMBL2404...)
Affinity DataIC50: 40nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029157(3-Piperidin-4-ylmethyl-1H-indole | CHEMBL429771)
Affinity DataIC50: 50nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029140(3-(3-Piperidin-4-yl-propyl)-1H-indole | CHEMBL2404...)
Affinity DataIC50: 60nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM77970(CLOMIPRAMINE HYDROCHLORIDE | CHLORIMIPRAMINE | 3-(...)
Affinity DataIC50: 70nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)
Affinity DataIC50: 100nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: 130nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029153(5-Methoxy-3-(2-piperidin-4-yl-ethyl)-1H-indole | C...)
Affinity DataIC50: 140nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50: 150nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)
Affinity DataIC50: 170nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: 220nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029151(1-Benzyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50: 300nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029142(1-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; fum...)
Affinity DataIC50: 400nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029143(1-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50: 400nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029143(1-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50: 400nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029152(3-[2-(1-Methyl-piperidin-4-yl)-ethyl]-1H-indole | ...)
Affinity DataIC50: 450nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029140(3-(3-Piperidin-4-yl-propyl)-1H-indole | CHEMBL2404...)
Affinity DataIC50: 500nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029157(3-Piperidin-4-ylmethyl-1H-indole | CHEMBL429771)
Affinity DataIC50: 550nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029145(3-(2-Piperidin-4-yl-ethyl)-1H-indol-5-ol; fumarate)
Affinity DataIC50: 600nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50: 600nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029148(5-Bromo-3-piperidin-4-ylmethyl-1H-indole | CHEMBL2...)
Affinity DataIC50: 600nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: 650nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029144(5-Chloro-3-piperidin-4-ylmethyl-1H-indole; 5 moles...)
Affinity DataIC50: 700nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029148(5-Bromo-3-piperidin-4-ylmethyl-1H-indole | CHEMBL2...)
Affinity DataIC50: 700nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM77970(CLOMIPRAMINE HYDROCHLORIDE | CHLORIMIPRAMINE | 3-(...)
Affinity DataIC50: 700nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029145(3-(2-Piperidin-4-yl-ethyl)-1H-indol-5-ol; fumarate)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029147(2-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029148(5-Bromo-3-piperidin-4-ylmethyl-1H-indole | CHEMBL2...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029142(1-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; fum...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029142(1-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; fum...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029149(2-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029155(5-Methoxy-3-piperidin-4-ylmethyl-1H-indole | CHEMB...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029156(1-Methyl-3-[2-(1-methyl-piperidin-4-yl)-ethyl]-1H-...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029144(5-Chloro-3-piperidin-4-ylmethyl-1H-indole; 5 moles...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM77970(CLOMIPRAMINE HYDROCHLORIDE | CHLORIMIPRAMINE | 3-(...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029151(1-Benzyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029153(5-Methoxy-3-(2-piperidin-4-yl-ethyl)-1H-indole | C...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029152(3-[2-(1-Methyl-piperidin-4-yl)-ethyl]-1H-indole | ...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029155(5-Methoxy-3-piperidin-4-ylmethyl-1H-indole | CHEMB...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029143(1-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029157(3-Piperidin-4-ylmethyl-1H-indole | CHEMBL429771)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029147(2-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50029150(CHEMBL276520 | 3-(2-Piperidin-4-yl-ethyl)-1H-indol...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
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