Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50048620
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50007422((R)-10,11-Dihydroxy-6-propyl-5,6,6a,7-tetrahydro-4...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50007422((R)-10,11-Dihydroxy-6-propyl-5,6,6a,7-tetrahydro-4...)
Affinity DataIC50: 5nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50010698((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223503(CHEMBL35556)
Affinity DataIC50: 24nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM52987(MLS000860063 | (R)-6-propyl-5,6,6a,7-tetrahydro-4H...)
Affinity DataIC50: 25nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50012987(CHEMBL553060 | 6-(2-Hydroxy-ethyl)-5,6,6a,7-tetrah...)
Affinity DataIC50: 25nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223517(CHEMBL285414)
Affinity DataIC50: 25nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223520(CHEMBL284248)
Affinity DataIC50: 30nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM84636(CHEMBL27559 | NPA-11-OH-R,(+))
Affinity DataIC50: 36nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223518(CHEMBL36061)
Affinity DataIC50: 112nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223519(CHEMBL32330)
Affinity DataIC50: 143nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223514(CHEMBL286929)
Affinity DataIC50: 204nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50007422((R)-10,11-Dihydroxy-6-propyl-5,6,6a,7-tetrahydro-4...)
Affinity DataIC50: 280nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223516(CHEMBL283871)
Affinity DataIC50: 394nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM52987(MLS000860063 | (R)-6-propyl-5,6,6a,7-tetrahydro-4H...)
Affinity DataIC50: 600nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50007422((R)-10,11-Dihydroxy-6-propyl-5,6,6a,7-tetrahydro-4...)
Affinity DataIC50: 670nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223513(CHEMBL440846)
Affinity DataIC50: 700nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM84636(CHEMBL27559 | NPA-11-OH-R,(+))
Affinity DataIC50: 700nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223503(CHEMBL35556)
Affinity DataIC50: 725nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 860nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223517(CHEMBL285414)
Affinity DataIC50: 900nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50016019(CHEMBL154709 | 10-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50010698((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223521(CHEMBL284368)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223520(CHEMBL284248)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223514(CHEMBL286929)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223516(CHEMBL283871)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50016019(CHEMBL154709 | 10-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223512(CHEMBL32392)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandPNGBDBM50223519(CHEMBL32330)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed