Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50041017
TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.631nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  4nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM22915(CHEMBL61618 | 5-[3-(benzyloxy)propyl]-1H-imidazole...)
Affinity DataKi:  20nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PDB3D3D Structure (crystal)
TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403581(CHEMBL291369)
Affinity DataKi:  20nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403575(CHEMBL59679)
Affinity DataKi:  25nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403577(CHEMBL443322)
Affinity DataKi:  25nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403578(CHEMBL60342)
Affinity DataKi:  25nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403580(CHEMBL62244)
Affinity DataKi:  79nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403576(CHEMBL59851)
Affinity DataKi:  126nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetHistamine H3 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403582(CHEMBL60606)
Affinity DataKi:  200nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article