Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50041010
LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  0.398nMAssay Description:Compound was tested for inhibiting [3H]pirenzepine Binding to Muscarinic receptor (M1) receptor in Rat Cortex HomogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  0.398nMAssay Description:Compound was tested for inhibiting [3H]pirenzepine Binding to Muscarinic receptor (M1) receptor in Rat Cortex HomogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50176065(CHEMBL76897 | CHEMBL168067 | 4-Diphenylacetoxy-1,1...)
Affinity DataKi:  0.513nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic acetylcholine receptor M4 in NG 108-15 CellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50176065(CHEMBL76897 | CHEMBL168067 | 4-Diphenylacetoxy-1,1...)
Affinity DataKi:  0.589nMAssay Description:Compound was tested for inhibiting [3H]pirenzepine Binding to Muscarinic receptor (M1) receptor in Rat Cortex HomogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50176065(CHEMBL76897 | CHEMBL168067 | 4-Diphenylacetoxy-1,1...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M3) in Rat Submaxillary GlandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403484(CHEMBL306182)
Affinity DataKi:  2.80nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M2) in Rat HeartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403484(CHEMBL306182)
Affinity DataKi:  3nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M3) in Rat Submaxillary GlandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50176065(CHEMBL76897 | CHEMBL168067 | 4-Diphenylacetoxy-1,1...)
Affinity DataKi:  4nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M2) in Rat HeartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  4.40nMAssay Description:Compound was tested for binding affinity against Muscarinic acetylcholine receptor M4 in NG 108-15 cell homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  4.70nMAssay Description:Compound was tested for binding affinity against Muscarinic acetylcholine receptor M4 in NG 108-15 cell homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403484(CHEMBL306182)
Affinity DataKi:  5nMAssay Description:Compound was tested for inhibiting [3H]pirenzepine Binding to Muscarinic receptor (M1) receptor in Rat Cortex HomogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  6.5nMAssay Description:Compound was tested for inhibiting [3H]pirenzepine Binding to Muscarinic receptor (M1) receptor in Rat Cortex HomogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  10nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M3) in Rat Submaxillary GlandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  10.5nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M3) in Rat Submaxillary GlandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403484(CHEMBL306182)
Affinity DataKi:  11nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic acetylcholine receptor M4 in NG 108-15 CellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  12nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M2) in Rat HeartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM50403485(CHEMBL292857)
Affinity DataKi:  33nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M2) in Rat HeartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  35nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic acetylcholine receptor M4 in NG 108-15 CellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  174nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M3) in Rat Submaxillary GlandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  794nMAssay Description:Compound was tested for inhibiting [3H]N-Methyl-scopolamine Binding to Muscarinic receptor (M2) in Rat HeartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article