Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50034902
LigandPNGBDBM50290469(5-[3-amino(imino)methylaminopropyl]-3-[1-cyclohexy...)
Affinity DataIC50: 25nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290477(N-(3-{1-[1-Cyclohexylmethyl-2-oxo-2-(4-phenyl-pipe...)
Affinity DataIC50: 30nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290463(N-[3-(1-{1-Cyclohexylmethyl-2-[4-(2,6-dimethyl-phe...)
Affinity DataIC50: 40nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290466(N-(3-{1-[1-Cyclohexylmethyl-2-oxo-2-(4-o-tolyl-pip...)
Affinity DataIC50: 40nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290470(N-[3-(1-{1-Cyclohexylmethyl-2-[4-(2,4-dimethyl-phe...)
Affinity DataIC50: 60nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50366479(CHEMBL1790511)
Affinity DataIC50: 200nMAssay Description:Tested for the ability to compete with [125I]-CO13 ([125I]-Y-F-K-A-Cha-G-L-dF-R) for binding to C5a anaphylatoxin chemotactic receptor from human neu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290463(N-[3-(1-{1-Cyclohexylmethyl-2-[4-(2,6-dimethyl-phe...)
Affinity DataIC50: 220nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290487(5-[3-amino(imino)methylaminopropyl]-3-[1-(4-fluoro...)
Affinity DataIC50: 230nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290481(5-[4-amino(imino)methylaminobutyl]-3-[1-cyclohexyl...)
Affinity DataIC50: 300nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290470(N-[3-(1-{1-Cyclohexylmethyl-2-[4-(2,4-dimethyl-phe...)
Affinity DataIC50: 300nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290469(5-[3-amino(imino)methylaminopropyl]-3-[1-cyclohexy...)
Affinity DataIC50: 300nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290476(5-[3-amino(imino)methylaminopropyl]-3-[1-cyclohexy...)
Affinity DataIC50: 300nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290466(N-(3-{1-[1-Cyclohexylmethyl-2-oxo-2-(4-o-tolyl-pip...)
Affinity DataIC50: 350nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290477(N-(3-{1-[1-Cyclohexylmethyl-2-oxo-2-(4-phenyl-pipe...)
Affinity DataIC50: 400nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290484(5-[3-amino(imino)methylaminopropyl]-3-[3-phenyl-1-...)
Affinity DataIC50: 450nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290465(5-[3-amino(imino)methylaminopropyl]-3-[3-methyl-1-...)
Affinity DataIC50: 450nMAssay Description:Tested for the ability to compete with [125I]-CO13 ([125I]-Y-F-K-A-Cha-G-L-dF-R) for binding to C5a anaphylatoxin chemotactic receptor from human neu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290467(CHEMBL70043 | CHEMBL71841 | 5-[3-amino(imino)methy...)
Affinity DataIC50: 800nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290475(5-(3-amino(imino)methylaminopropyl)-3-(1-(2-naphth...)
Affinity DataIC50: 900nMAssay Description:Tested for the its ability to compete with [125I]-CO13 [125I]-Y-F-K-A-Cha-G-L-dF-R) for binding to C5a anaphylatoxin chemotactic receptor of human ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290479(N-(3-{1-[1-Cyclohexylmethyl-2-oxo-2-(4-phenyl-pipe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50366479(CHEMBL1790511)
Affinity DataIC50: 1.20E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290480(5-[3-amino(imino)methylaminopropyl]-3-[2-methyl-1-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290476(5-[3-amino(imino)methylaminopropyl]-3-[1-cyclohexy...)
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290483(5-[3-amino(imino)methylaminopropyl]-3-[1-cyclohexy...)
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290465(5-[3-amino(imino)methylaminopropyl]-3-[3-methyl-1-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290473(5-[3-amino(imino)methylaminopropyl]-3-[1-(2-naphth...)
Affinity DataIC50: 2.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290475(5-(3-amino(imino)methylaminopropyl)-3-(1-(2-naphth...)
Affinity DataIC50: 2.30E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290464(5-[3-amino(imino)methylaminopropyl]-3-[1-spiro[2,3...)
Affinity DataIC50: 3.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290474(5-[3-amino(imino)methylaminopropyl]-3-[3-phenyl-1-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290482(5-[3-amino(imino)methylaminopropyl]-3-[3-methylsul...)
Affinity DataIC50: 3.40E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290485(5-[3-amino(imino)methylaminopropyl]-3-[1-(4-hydrox...)
Affinity DataIC50: 4.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290468(5-(4-aminobutyl)-3-[1-cyclohexylmethyl-2-oxo-2-spi...)
Affinity DataIC50: 4.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290467(CHEMBL70043 | CHEMBL71841 | 5-[3-amino(imino)methy...)
Affinity DataIC50: 4.00E+3nMAssay Description:Tested for the ability to compete with [125I]-CO13 ([125I]-Y-F-K-A-Cha-G-L-dF-R) for binding to C5a anaphylatoxin chemotactic receptor from human neu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290478(5-[3-amino(imino)methylaminopropyl]-3-[1-(4-cycloh...)
Affinity DataIC50: 5.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290484(5-[3-amino(imino)methylaminopropyl]-3-[3-phenyl-1-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290467(CHEMBL70043 | CHEMBL71841 | 5-[3-amino(imino)methy...)
Affinity DataIC50: 8.00E+3nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50290486(5-[3-amino(imino)methylaminopropyl]-3-[1-(1-naphth...)
Affinity DataIC50: 1.10E+4nMAssay Description:Tested for its ability to compete with [125I]C5a for binding to C5a anaphylatoxin chemotactic receptor of human neutrophil membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article