Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50030134
LigandPNGBDBM50291452(N-Methyl-N'-(6-phenethyloxy-biphenyl-3-yl)-guanidi...)
Affinity DataIC50: 800nMAssay Description:Compound was evaluated for the antagonistic activity against C5a anaphylatoxin chemotactic receptor in human neutrophil C5a stimulated respiratory bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291461(N-Methyl-N'-[6-(3-phenyl-propoxy)-biphenyl-3-yl]-g...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291465(N-[6-(2-Cyclohexyl-ethoxy)-biphenyl-3-yl]-N'-methy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291456(N-(6-Benzyloxy-biphenyl-3-yl)-N'-methyl-guanidine ...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291460(N-(6-Cyclohexylmethoxy-biphenyl-3-yl)-N'-methyl-gu...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291468(N-(4-Benzyloxy-3-phenoxy-phenyl)-N'-methyl-guanidi...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291467(N-[3-Benzyloxy-4-(4-phenyl-butoxy)-phenyl]-N'-meth...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291470(N-(4-Benzyloxy-3-naphthalen-1-yl-phenyl)-N'-methyl...)
Affinity DataIC50: 4.50E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291453(N-[3-Benzyloxy-4-(3-phenyl-propoxy)-phenyl]-N'-met...)
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291466(N-(3-Benzyloxy-4-phenethyloxy-phenyl)-N'-methyl-gu...)
Affinity DataIC50: 7.50E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291463(N-(3-Benzyloxy-4-cyclohexylmethoxy-phenyl)-N'-meth...)
Affinity DataIC50: 8.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291458(N-(6-Benzyloxy-3'-fluoro-biphenyl-3-yl)-N'-methyl-...)
Affinity DataIC50: 8.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291451(N-(6-Benzyloxy-3'-methoxy-biphenyl-3-yl)-N'-methyl...)
Affinity DataIC50: 9.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291469(N-[3-Benzyloxy-4-(2-cyclohexyl-ethoxy)-phenyl]-N'-...)
Affinity DataIC50: 9.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291462(N-(4-Benzyloxy-3-thiophen-2-yl-phenyl)-N'-methyl-g...)
Affinity DataIC50: 9.00E+3nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291464(N-(4-Benzyloxy-3-cyclopentyloxy-phenyl)-N'-methyl-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291455(N-(3-Benzyloxy-4-butoxy-phenyl)-N'-methyl-guanidin...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291457(N-(3,4-Bis-benzyloxy-phenyl)-N'-methyl-guanidine |...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291450(N-(6-Benzyloxy-4'-chloro-biphenyl-3-yl)-N'-methyl-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291459(N-(6-Benzyloxy-4'-methoxy-biphenyl-3-yl)-N'-methyl...)
Affinity DataIC50: 5.40E+4nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291454(N-(3,4-Bis-benzyloxy-phenyl)-guanidine | CHEMBL170...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity against C5a anaphylatoxin chemotactic receptor assayed on human monocyte cell line U937More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article