Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50030120
TargetVasopressin V2 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataIC50: 3.30nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 uM in LLCPKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V2 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50: 9.5nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 uM in LLCPKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50: 9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataIC50: 10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article