Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50029963
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289727(4-Hydroxy-piperidine-1-carboxylic acid ((S)-1-{[(S...)
Affinity DataIC50: 0.680nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289726(1H-Benzoimidazole-2-carboxylic acid [(S)-1-((1S,2S...)
Affinity DataIC50: 13nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 42nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 45nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of human plasma, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289716(5-Fluoro-1H-indole-2-carboxylic acid [(S)-1-((1S,2...)
Affinity DataIC50: 46nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289724(1-Oxo-1,2-dihydro-isoquinoline-3-carboxylic acid [...)
Affinity DataIC50: 48nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 93nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of monkey plasma, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289723(Benzofuran-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-...)
Affinity DataIC50: 140nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289720(5-Chloro-1H-indole-2-carboxylic acid [(S)-1-((1S,2...)
Affinity DataIC50: 260nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289722(1-Acetyl-1H-indole-2-carboxylic acid [(S)-1-((1S,2...)
Affinity DataIC50: 340nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289721((S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataIC50: 420nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289718(5-Hydroxy-1H-indole-2-carboxylic acid [(S)-1-((1S,...)
Affinity DataIC50: 600nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289725(Isoquinoline-3-carboxylic acid [(S)-1-((1S,2S,4S)-...)
Affinity DataIC50: 790nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289715(1H-Pyrrolo[2,3-b]pyridine-2-carboxylic acid [(S)-1...)
Affinity DataIC50: 800nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289713(2,3-Dihydro-1H-indole-2-carboxylic acid [(S)-1-((1...)
Affinity DataIC50: 880nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of human plasma, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289713(2,3-Dihydro-1H-indole-2-carboxylic acid [(S)-1-((1...)
Affinity DataIC50: 880nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289719(1H-Pyrrole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of dog plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289717(Benzo[b]thiophene-2-carboxylic acid [(S)-1-((1S,2S...)
Affinity DataIC50: 8.20E+3nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of marmoset plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetCathepsin D(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against cathepsin D (bovine), expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetRenin(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of rat plasma renin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetPepsin A(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory effect was evaluated against pepsin, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

TargetAngiotensin-converting enzyme(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289714(1H-Indole-2-carboxylic acid [(S)-1-((1S,2S,4S)-1-c...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against ACE human, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article