Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50029865
TargetDihydrofolate reductase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288820(LY-298207 | (S)-2-{(S)-4-[4-(2,4-Diamino-pyrimidin...)
Affinity DataKi:  0.00500nMAssay Description:Binding affinity against Recombinant human dihydrofolate reductase (DHFR)More data for this Ligand-Target Pair
In DepthDetails Article

TargetDihydrofolate reductase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288821((S)-2-{(S)-4-[3-(2,4-Diamino-pyrimidin-5-yl)-propy...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against Recombinant human dihydrofolate reductase (DHFR)More data for this Ligand-Target Pair
In DepthDetails Article

TargetThymidylate synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288820(LY-298207 | (S)-2-{(S)-4-[4-(2,4-Diamino-pyrimidin...)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against Recombinant human thymidylate synthase (TS).More data for this Ligand-Target Pair
In DepthDetails Article

TargetThymidylate synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288821((S)-2-{(S)-4-[3-(2,4-Diamino-pyrimidin-5-yl)-propy...)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against Recombinant human thymidylate synthase (TS)More data for this Ligand-Target Pair
In DepthDetails Article