Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50029836
LigandPNGBDBM50288501(2-{2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta...)
Affinity DataIC50: 660nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288479(8-Chloro-11-(1-phenylmethanesulfonyl-piperidin-4-y...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288481(8-Chloro-11-(1-ethenesulfonyl-piperidin-4-ylidene)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288506([(R)-2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohep...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288498(8-Chloro-11-(1-methanesulfonyl-piperidin-4-ylidene...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288495(4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,2-b...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288499(2-{2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288507([(S)-2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohep...)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288502(2-[(R)-2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288478(2-{(R)-2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288480(2-{(R)-1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288505((R)-5-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohept...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288500(11-[1-(Butane-1-sulfonyl)-piperidin-4-ylidene]-8-c...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288491(8-Chloro-11-(1-ethanesulfonyl-piperidin-4-ylidene)...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288509((S)-2-Amino-1-[4-(8-chloro-5,6-dihydro-benzo[5,6]c...)
Affinity DataIC50: 6.29E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288493({2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1...)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288490(1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288504(N-{2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288497({2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288487(N-{2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta...)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288492(2-Benzylamino-1-[4-(8-chloro-5,6-dihydro-benzo[5,6...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288482(1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288508(2-{(R)-1-Benzyl-2-[4-(8-chloro-5,6-dihydro-benzo[5...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288489(2-{(R)-1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288483(2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288486(2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288488(1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288485(8-Chloro-11-[1-(octane-1-sulfonyl)-piperidin-4-yli...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288484(8-Chloro-11-[1-(4-nitro-benzenesulfonyl)-piperidin...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288494(8-Chloro-11-[1-(naphthalene-2-sulfonyl)-piperidin-...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288496(8-Chloro-11-[1-(thiophene-2-sulfonyl)-piperidin-4-...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50288503(2-Amino-1-[4-(8-chloro-5,6-dihydro-benzo[5,6]cyclo...)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article