Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50029796
TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287969((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50: 0.100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287978((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50: 0.100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287967((S)-3-Benzo[1,3]dioxol-5-yl-3-{[(R)-1-(3-piperidin...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287983(5-Methyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287982(3-{[1-(3-Piperazin-1-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287972(2-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083463((R)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287985(3-Phenyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083467((S)-5-Phenyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287977(3-{[(S)-1-(3-Piperidin-4-yl-propionyl)-piperidine-...)
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083459(2-Hydroxy-3-{[(R)-1-(3-piperidin-4-yl-propionyl)-p...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50034703(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083452(3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperidine-...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287973(3-({1-[3-(1-Methyl-piperidin-4-yl)-propionyl]-pipe...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287981(3-{[1-(3-Piperidin-4-yl-propionyl)-pyrrolidine-3-c...)
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287970(4-Oxo-1-[1-(3-piperidin-4-yl-propionyl)-piperidine...)
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287980(3-{[1-(3-Piperidin-4-yl-propionyl)-azepane-3-carbo...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287978((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287967((S)-3-Benzo[1,3]dioxol-5-yl-3-{[(R)-1-(3-piperidin...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287976(3-({1-[(Piperidin-4-ylmethyl)-carbamoyl]-piperidin...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287965(3-(2-Carboxy-ethylcarbamoyl)-piperidine-1-carboxyl...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287979(3-{[1-(2-Piperidin-4-yl-ethanesulfonyl)-piperidine...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083476((S)-6,6-Dimethyl-3-{[(R)-1-(3-piperidin-4-yl-propi...)
Affinity DataIC50: 21nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083476((S)-6,6-Dimethyl-3-{[(R)-1-(3-piperidin-4-yl-propi...)
Affinity DataIC50: 80nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083467((S)-5-Phenyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl...)
Affinity DataIC50: 80nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287969((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287966(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-4-ca...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287984(2-Methyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287968(2-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287971(3-{Methyl-[1-(3-piperidin-4-yl-propionyl)-piperidi...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083452(3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperidine-...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287974(1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbox...)
Affinity DataIC50: 600nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50034703(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083459(2-Hydroxy-3-{[(R)-1-(3-piperidin-4-yl-propionyl)-p...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287972(2-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287973(3-({1-[3-(1-Methyl-piperidin-4-yl)-propionyl]-pipe...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50083463((R)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287977(3-{[(S)-1-(3-Piperidin-4-yl-propionyl)-piperidine-...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287985(3-Phenyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287983(5-Methyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287965(3-(2-Carboxy-ethylcarbamoyl)-piperidine-1-carboxyl...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287981(3-{[1-(3-Piperidin-4-yl-propionyl)-pyrrolidine-3-c...)
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287976(3-({1-[(Piperidin-4-ylmethyl)-carbamoyl]-piperidin...)
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287980(3-{[1-(3-Piperidin-4-yl-propionyl)-azepane-3-carbo...)
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287982(3-{[1-(3-Piperazin-1-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287984(2-Methyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287966(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-4-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287968(2-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287979(3-{[1-(2-Piperidin-4-yl-ethanesulfonyl)-piperidine...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProteinase-activated receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287971(3-{Methyl-[1-(3-piperidin-4-yl-propionyl)-piperidi...)
Affinity DataIC50: 2.80E+4nMAssay Description:In vitro inhibition of thrombin-induced human gel-filtered platelet aggregation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

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