Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50029726
LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50: 130nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50: 2.70E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50: 2.70E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50: 3.35E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50: 4.36E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50: 4.47E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50: 5.50E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50: 6.32E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50: 6.69E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50: 7.57E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50: 7.82E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50: 8.09E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50: 8.09E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50: 8.10E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50: 8.76E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50: 9.44E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50: 3.23E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50: 2.90E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50: 2.04E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50: 7.21E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article