Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50029691
LigandPNGBDBM50286892(1-[(R)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.0700nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286884(1-{1-[2-(1-Methyl-cyclopentyl)-2-oxo-ethyl]-2-oxo-...)
Affinity DataIC50: 0.100nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.230nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286886(1-[1-(3-Cyclohexyl-2-oxo-propyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 0.280nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286888(1-{1-[2-(1-Methyl-cyclohexyl)-2-oxo-ethyl]-2-oxo-5...)
Affinity DataIC50: 0.380nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286891(1-[1-(2-Cyclohexyl-2-oxo-ethyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50: 0.400nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286885(1-{1-[2-(1-Methyl-cyclopropyl)-2-oxo-ethyl]-2-oxo-...)
Affinity DataIC50: 0.410nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.520nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286883(1-[1-(3,3-Dimethyl-2-oxo-pentyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 0.570nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286889(1-[1-(3-Cyclohexyl-3-methyl-2-oxo-butyl)-2-oxo-5-p...)
Affinity DataIC50: 0.860nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286887(1-[1-(3-Ethyl-2-oxo-pentyl)-2-oxo-5-phenyl-2,3-dih...)
Affinity DataIC50: 1.90nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286890(1-[1-(2-Cycloheptyl-2-oxo-ethyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 2nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286881(1-[1-(3-Methyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3-dih...)
Affinity DataIC50: 2.10nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286893(1-[1-(2-Cyclobutyl-2-oxo-ethyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50: 2.40nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 6.10nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 111nMAssay Description:Compound was evaluated for its ability to displace [3H]L-364718 from Cholecystokinin type A receptor from rat pancreas at dose of 0.03 umol/kgMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 146nMAssay Description:Compound was evaluated for its ability to displace [3H]L-364718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286884(1-{1-[2-(1-Methyl-cyclopentyl)-2-oxo-ethyl]-2-oxo-...)
Affinity DataIC50: 293nMAssay Description:Compound was evaluated for its ability to displace [3H]-L-364,718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286892(1-[(R)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 440nMAssay Description:Compound was evaluated for its ability to displace [3H]-L-364,718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286886(1-[1-(3-Cyclohexyl-2-oxo-propyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 480nMAssay Description:Compound was evaluated for its ability to displace [3H]-L-364,718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286883(1-[1-(3,3-Dimethyl-2-oxo-pentyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 720nMAssay Description:Compound was evaluated for its ability to displace [3H]-L-364,718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286881(1-[1-(3-Methyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3-dih...)
Affinity DataIC50: 1.20E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]-L-364,718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 2.50E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]-L-364,718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286888(1-{1-[2-(1-Methyl-cyclohexyl)-2-oxo-ethyl]-2-oxo-5...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was evaluated for its ability to displace [3H]-L-364,718 from Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article