Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50029646
TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286537(3-{[1-Oxo-2-(2-piperidin-4-yl-ethyl)-1,2,3,4-tetra...)
Affinity DataIC50: 79nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286527(3-{[1-Oxo-2-(2-piperidin-4-yl-ethyl)-2,3,4,5-tetra...)
Affinity DataIC50: 170nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286535(3-{[8-Methyl-1-oxo-2-(2-piperidin-4-yl-ethyl)-1,2,...)
Affinity DataIC50: 170nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50058238(CHEMBL540024 | CHEMBL288521 | 3-{[4-Oxo-5-(2-piper...)
Affinity DataIC50: 250nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50058240(3-{[4-Oxo-5-(2-piperidin-4-yl-ethyl)-5,6,7,8-tetra...)
Affinity DataIC50: 470nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286531(3-{[9-Methyl-1-oxo-2-(2-piperidin-4-yl-ethyl)-2,3,...)
Affinity DataIC50: 510nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286534(3-{[4-Oxo-5-(3-piperidin-4-yl-propyl)-4,5,6,7-tetr...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286536({[4-Oxo-5-(3-piperidin-4-yl-propyl)-4,5,6,7-tetrah...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286532(4-[(4-Oxo-5-piperidin-4-ylmethyl-4,5,6,7-tetrahydr...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50241180(3-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286530(3-[4-Oxo-2-(2-piperidin-4-yl-ethylcarbamoyl)-6,7-d...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286533(3-[(4-Oxo-5-piperidin-4-ylmethyl-4,5,6,7-tetrahydr...)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286529(3-{[1-Oxo-9-phenyl-2-(2-piperidin-4-yl-ethyl)-2,3,...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of fibrinogen binding to glycoprotein alpha IIb beta-3 integrin of activated plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article