Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50029569
TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285678((1-{(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 0.380nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285677((1-{(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285683((1-{(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285675((1-{(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 0.650nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285671({1-[(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285674((1-{(R)-1-{3-[(E)-2-(2,3-Difluoro-thieno[3,2-b]pyr...)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285670((1-{(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 1.05nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285672((1-{(R)-1-{3-[2-(2,3-Dichloro-thieno[3,2-b]pyridin...)
Affinity DataIC50: 1.06nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285673((1-{(R)-1-{3-[(E)-2-(2-Chloro-thieno[3,2-b]pyridin...)
Affinity DataIC50: 1.16nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285676([1-((R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 1.63nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285682((1-{(R)-1-{3-[(E)-2-(3-Chloro-thieno[3,2-b]pyridin...)
Affinity DataIC50: 1.91nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285680((1-{(R)-1-[3-(2,3-Dichloro-thieno[3,2-b]pyridin-5-...)
Affinity DataIC50: 2.01nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285686({1-[(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 2.16nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285679([1-((R)-3-(2-Bromo-phenyl)-1-{3-[(E)-2-(2,3-dichlo...)
Affinity DataIC50: 2.43nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285685({1-[(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 3.36nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285681([1-((R)-3-(4-Bromo-phenyl)-1-{3-[(E)-2-(2,3-dichlo...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285688((1-{(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 6.42nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285684((1-{(R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 8.49nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285669({1-[(R)-1-{3-[(E)-2-(2,3-Dichloro-thieno[3,2-b]pyr...)
Affinity DataIC50: 8.67nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285689((1-{(R)-1-{3-[2-(2,3-Dichloro-thieno[3,2-b]pyridin...)
Affinity DataIC50: 15.7nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285687((1-{(R)-1-[3-(2,3-Dichloro-thieno[3,2-b]pyridin-5-...)
Affinity DataIC50: 150nMAssay Description:Inhibition of binding of [ H]-LTD4 to DMSO differentiated U937 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article