Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50029482
TargetMu-type opioid receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataKd:  0.400nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO expressed as KdMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetMu-type opioid receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50030143(bis-(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azape...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO expressed as KdMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetMu-type opioid receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataIC50: 1.40nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO expressed as KdMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetMu-type opioid receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50284914(MET-TAMO and N-CPM-MET-TAMO analogue | CHEMBL29760...)
Affinity DataIC50: 2.90nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO expressed as KdMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetMu-type opioid receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50030145(bis-(1N-[4-cyclopropylmethyl-10-hydroxy-14-oxo-12-...)
Affinity DataIC50: 3.90nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO expressed as KdMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataIC50: 5.30nMAssay Description:Inhibitory activity against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataIC50: 7.70nMAssay Description:Inhibitory activity against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50030145(bis-(1N-[4-cyclopropylmethyl-10-hydroxy-14-oxo-12-...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50030143(bis-(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azape...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50030145(bis-(1N-[4-cyclopropylmethyl-10-hydroxy-14-oxo-12-...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50030143(bis-(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azape...)
Affinity DataIC50: 41nMAssay Description:Inhibitory activity against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284914(MET-TAMO and N-CPM-MET-TAMO analogue | CHEMBL29760...)
Affinity DataIC50: 52nMAssay Description:Inhibitory activity against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284914(MET-TAMO and N-CPM-MET-TAMO analogue | CHEMBL29760...)
Affinity DataIC50: 89nMAssay Description:Inhibitory activity against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article