Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029454
TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284686((3S,4S)-6-(6-Methyl-5-nitro-pyridin-2-ylmethoxy)-3...)
Affinity DataKi:  240nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284685((3S,4S)-6-(5-Bromo-6-methyl-pyridin-2-ylmethoxy)-3...)
Affinity DataKi:  1.56E+3nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284680(3-Pyridin-3-ylmethyl-6-(quinolin-2-ylmethoxy)-chro...)
Affinity DataKi:  1.64E+3nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50012434(1-[3-(Quinolin-2-ylmethoxy)-phenyl]-hexan-1-ol | 1...)
Affinity DataKi:  8.00E+3nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284683((3S,4S)-6-(6-Chloro-pyridin-2-ylmethoxy)-3-pyridin...)
Affinity DataKi:  2.34E+4nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284688((3S,4S)-6-(Pyridin-2-ylmethoxy)-3-pyridin-3-ylmeth...)
Affinity DataKi: >1.00E+5nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284684((3S,4S)-6-(6-Methyl-pyridin-2-ylmethoxy)-3-pyridin...)
Affinity DataKi: >1.00E+5nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284687((3S,4S)-6-(6-Fluoro-pyridin-2-ylmethoxy)-3-pyridin...)
Affinity DataKi: >1.00E+5nMAssay Description:Compound was tested for the inhibition of [3H]leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article