Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029218
TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282359(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: 0.800nMAssay Description:In vitro binding affinity evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II receptor, type 1 i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282358(N-[4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II receptor, type 1 i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282360(2-Ethyl-6,8-dimethyl-3-[2'-(2H-tetrazol-5-yl)-biph...)
Affinity DataIC50: 5.70nMAssay Description:In vitro binding affinity evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II receptor, type 1 i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282358(N-[4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282359(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282360(2-Ethyl-6,8-dimethyl-3-[2'-(2H-tetrazol-5-yl)-biph...)
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity at AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from rat brain memb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282361(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282361(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: 83nMAssay Description:In vitro binding affinity evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II receptor, type 1 i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article