Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50029213
TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282309(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50009718(CHEMBL7550 | 2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetraz...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282310(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50281848(L-158827 | 2-Ethyl-5,7-dimethyl-3-{4-[2-(2H-tetraz...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 3nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282307(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282306(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282305(5-Ethyl-3-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]p...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282311(5-Benzyl-3-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282308(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 22nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282308(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 24nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281848(L-158827 | 2-Ethyl-5,7-dimethyl-3-{4-[2-(2H-tetraz...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50009718(CHEMBL7550 | 2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetraz...)
Affinity DataIC50: 37nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282304(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 44nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282312(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 87nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282312(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 120nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282307(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 130nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282311(5-Benzyl-3-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]...)
Affinity DataIC50: 150nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282306(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 150nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282304(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 190nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282305(5-Ethyl-3-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]p...)
Affinity DataIC50: 900nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282309(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282310(3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of rat midbrain angiotensin II type 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article