Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50029079
LigandPNGBDBM50281270(Acetic acid (2S,3S)-5-(2-dimethylamino-ethyl)-8-me...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50281272((2R,3S)-5-(2-Dimethylamino-ethyl)-8-methoxy-2-(4-m...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50004704(Acetic acid 5-(2-dimethylamino-ethyl)-2-(4-methoxy...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50281271((2R,3S)-5-(2-Dimethylamino-ethyl)-2-(4-methoxy-phe...)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50000383(CHEMBL98189 | 1-(2-Dimethylamino-ethyl)-4-(4-metho...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel of guinea pig striated muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article