Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50029035
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 10nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 18nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 20nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280871(12-(3-azidopropyl)-13-methyl-6,7,12,13-tetrahydro-...)
Affinity DataIC50: 25nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280873(2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...)
Affinity DataIC50: 27nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280870(12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...)
Affinity DataIC50: 32nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 40nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280877(2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 75nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280875(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 82nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280868(12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...)
Affinity DataIC50: 99nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280869(13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo...)
Affinity DataIC50: 100nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280875(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 110nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: 200nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280868(12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...)
Affinity DataIC50: 280nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280877(2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 320nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280868(12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...)
Affinity DataIC50: 390nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280876(12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 400nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280870(12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...)
Affinity DataIC50: 440nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280871(12-(3-azidopropyl)-13-methyl-6,7,12,13-tetrahydro-...)
Affinity DataIC50: 450nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280878(12,13-dimethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-...)
Affinity DataIC50: 450nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280877(2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 500nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280876(12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 520nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280874(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 590nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 650nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 680nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: 700nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280870(12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...)
Affinity DataIC50: 710nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280876(12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280873(2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280873(2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280874(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280870(12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...)
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50212623(CHEMBL299248)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280868(12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...)
Affinity DataIC50: 4.80E+3nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280869(13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo...)
Affinity DataIC50: 5.10E+3nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280878(12,13-dimethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-...)
Affinity DataIC50: 5.50E+3nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280878(12,13-dimethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-...)
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

TargetcGMP-dependent protein kinase 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 6.20E+3nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280873(2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...)
Affinity DataIC50: 6.30E+3nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50212624(CHEMBL294684)
Affinity DataIC50: 8.10E+3nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280877(2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280876(12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280867(2-(6,13-dimethyl-5-oxo-6,7,12,13-tetrahydro-5H-ind...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50280869(13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo...)
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article

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