Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50029002
TargetSerine protease 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280654((S)-5-Guanidino-2-{[(S)-1-((S)-2-methylamino-2-phe...)
Affinity DataIC50: 20nMAssay Description:In vitro concentration of compound required to inhibit 50% of trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProthrombin(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280654((S)-5-Guanidino-2-{[(S)-1-((S)-2-methylamino-2-phe...)
Affinity DataIC50: 20nMAssay Description:In vitro concentration of compound required to inhibit 50% of 6 nM thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProthrombin(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280655(3-Isobutyryloxy-benzo[4,5]thieno[3,2-b]furan-2-car...)
Affinity DataIC50: 30nMAssay Description:In vitro concentration of compound required to inhibit 50% of 6 nM thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCoagulation factor X(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280655(3-Isobutyryloxy-benzo[4,5]thieno[3,2-b]furan-2-car...)
Affinity DataIC50: 100nMAssay Description:In vitro concentration of compound required to inhibit 50% of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetPlasminogen(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280654((S)-5-Guanidino-2-{[(S)-1-((S)-2-methylamino-2-phe...)
Affinity DataIC50: 500nMAssay Description:In vitro concentration of compound required to inhibit 50% of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCoagulation factor X(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280654((S)-5-Guanidino-2-{[(S)-1-((S)-2-methylamino-2-phe...)
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro concentration of compound required to inhibit 50% of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280655(3-Isobutyryloxy-benzo[4,5]thieno[3,2-b]furan-2-car...)
Affinity DataIC50: 7.20E+3nMAssay Description:In vitro concentration of compound required to inhibit 50% of KallikreinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProthrombin(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280656(3-Hydroxy-benzo[4,5]thieno[3,2-b]furan-2-carboxyli...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro concentration of compound required to inhibit 50% of 6 nM thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProthrombin(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280657(3-Dimethylcarbamoyloxy-benzo[4,5]thieno[3,2-b]fura...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro concentration of compound required to inhibit 50% of 6 nM thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProthrombin(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280658(3-Methoxy-benzo[4,5]thieno[3,2-b]furan-2-carboxyli...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro concentration of compound required to inhibit 50% of 6 nM thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280654((S)-5-Guanidino-2-{[(S)-1-((S)-2-methylamino-2-phe...)
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro concentration of compound required to inhibit 50% of kallikreinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetSerine protease 1(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50280655(3-Isobutyryloxy-benzo[4,5]thieno[3,2-b]furan-2-car...)
Affinity DataIC50: 2.90E+4nMAssay Description:In vitro concentration of compound required to inhibit 50% of trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetPlasminogen(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280655(3-Isobutyryloxy-benzo[4,5]thieno[3,2-b]furan-2-car...)
Affinity DataIC50: 2.40E+5nMAssay Description:In vitro concentration of compound required to inhibit 50% of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article